SCHEMBL6996630

SCHEMBL6996630

COc1c(C)cc(C2=C(c3ccc(S(N)(=O)=O)cc3)OC(C)(C)C2=O)cc1C

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.45
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
CA9 Q16790 2/20 0.45
PTGS2 P35354 15/20 0.42
PTGS1 P23219 8/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6993170 0.89 CA1 (0.60) CA12CA1CA2CA9PTGS2
SCHEMBL6993196 0.89 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL6999644 0.85 PTGS2 (0.49) CA12CA1CA2CA9PTGS2
SCHEMBL6998922 0.83 PTGS2 (0.51) CA12CA1CA2CA9PTGS2
SCHEMBL7004184 0.81 PTGS2 (0.46) PTGS2PTGS1
SCHEMBL7000063 0.81 PTGS2 (0.45) CA12CA1CA2CA9PTGS2
SCHEMBL7002045 0.81 CA9 (0.52) CA12CA1CA2CA9PTGS2
SCHEMBL6999688 0.81 PTGS2 (0.60) CA12CA1CA2CA9PTGS2
SCHEMBL7000979 0.81 PTGS2 (0.48) CA12CA1CA2CA9PTGS2
SCHEMBL7002002 0.80 PTGS2 (0.56) CA12CA1CA2CA9PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109799-B1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORP (KR) 2003-12-17 EP claimed
US-6492416-B1 TREATING INFLAMMATION AND ASSOCIATED DISORDERS PACIFIC CORPORATION (KR) 2002-12-10 US claimed
EP-1109799-B1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORP (KR) 2003-12-17 EP disclosed
US-6492416-B1 TREATING INFLAMMATION AND ASSOCIATED DISORDERS PACIFIC CORPORATION (KR) 2002-12-10 US disclosed