SCHEMBL7002045

SCHEMBL7002045

COc1cccc(C2=C(c3ccc(S(N)(=O)=O)cc3)OC(C)(C)C2=O)c1

nearest known ligand 0.72

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 8/20 0.52
CA2 P00918 7/20 0.52
CA1 P00915 5/20 0.48
CA4 P22748 1/20 0.48
CA5A P35218 1/20 0.48
CA5B Q9Y2D0 1/20 0.48
PTGS2 P35354 3/20 0.46
CA12 O43570 4/20 0.45
PGR P06401 1/20 0.44
CDK1 P06493 1/20 0.43
CDK2 P24941 1/20 0.43
ALKBH3 Q96Q83 1/20 0.42
FAAH O00519 1/20 0.41
NAAA Q02083 1/20 0.41
CA7 P43166 1/20 0.40
CA14 Q9ULX7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6999220 0.90 PTGS2 (0.49) PTGS2PGRALKBH3
SCHEMBL7002517 0.87 CA9 (0.48) CA9CA2CA1CA4CA5A
SCHEMBL6999849 0.86 CA2 (0.53) CA9CA2CA1CA5ACA5B
SCHEMBL6999323 0.85 CA2 (0.54) CA9CA2CA1CA4CA5A
SCHEMBL7001251 0.85 CA2 (0.56) CA9CA2CA1CA4PTGS2
Polmacoxib SCHEMBL29351757 0.84 PTGS2 (0.55) CA9CA2CA1PTGS2CA12
SCHEMBL3232569 0.84 CA2 (0.51) CA9CA2CA1PTGS2CA12
SCHEMBL6998922 0.84 PTGS2 (0.51) CA9CA2CA1CA4PTGS2
Polmacoxib SCHEMBL3233093 0.84 PTGS2 (0.55) CA9CA2CA1PTGS2CA12
SCHEMBL7002002 0.83 PTGS2 (0.56) CA9CA2CA1CA4CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109799-B1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORP (KR) 2003-12-17 EP claimed
US-6492416-B1 TREATING INFLAMMATION AND ASSOCIATED DISORDERS PACIFIC CORPORATION (KR) 2002-12-10 US claimed
EP-1109799-A1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORPORATION (KR) 2001-06-27 EP claimed
WO-2000061571-A1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORPORATION (KR) 2000-10-19 WO claimed
EP-1109799-B1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORP (KR) 2003-12-17 EP disclosed
US-6492416-B1 TREATING INFLAMMATION AND ASSOCIATED DISORDERS PACIFIC CORPORATION (KR) 2002-12-10 US disclosed
EP-1109799-A1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORPORATION (KR) 2001-06-27 EP disclosed
WO-2000061571-A1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORPORATION (KR) 2000-10-19 WO disclosed