SCHEMBL6996829

SCHEMBL6996829

COc1ccc(CC(=O)N[C@H](C(=O)O)C(C)C)c(C)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
MAPK1 P28482 1/20 0.45
THRA P10827 3/20 0.45
THRB P10828 3/20 0.45
CASP1 P29466 2/20 0.45
CASP3 P42574 2/20 0.45
CASP7 P55210 2/20 0.45
CASP8 Q14790 2/20 0.45
NPSR1 Q6W5P4 1/20 0.44
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MMP9 P14780 2/20 0.42
MMP1 P03956 1/20 0.42
MMP2 P08253 1/20 0.42
MMP3 P08254 1/20 0.42
MMP7 P09237 1/20 0.42
MMP8 P22894 1/20 0.42
MMP13 P45452 1/20 0.42
AKR1C3 P42330 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6996825 1.00 MEN1 (0.47) MEN1KMT2AMAPK1THRATHRB
SCHEMBL7958352 0.90 ALDH1A1 (0.53) MEN1KMT2ATHRBCASP1CASP3
SCHEMBL6988661 0.90 ALDH1A1 (0.53) MEN1KMT2ATHRBCASP1CASP3
SCHEMBL6996018 0.89 KMT2A (0.47) MEN1KMT2AALDH1A1AKR1C3AKR1C2
SCHEMBL6996015 0.89 KMT2A (0.47) MEN1KMT2AALDH1A1AKR1C3AKR1C2
SCHEMBL6994002 0.86 SMN1; SMN2 (0.50) MEN1KMT2AALDH1A1KDM4E
SCHEMBL6994008 0.86 SMN1; SMN2 (0.50) MEN1KMT2AALDH1A1KDM4E
SCHEMBL4428330 0.86 PRSS1 (0.47) MEN1KMT2AMAPK1THRATHRB
SCHEMBL4428332 0.86 PRSS1 (0.47) MEN1KMT2AMAPK1THRATHRB
SCHEMBL7000904 0.83 ALDH1A1 (0.53) MEN1KMT2AMAPK1ALDH1A1MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0754175-B1 ALKOXY-ALKYL-SUBSTITUTED 1-H-3-ARYL-PYRROLIDINE-2,4-DIONES USED AS HERBICIDES AND PESTICIDES BAYER CROPSCIENCE AG (DE) 2003-01-29 EP disclosed
US-6172255-B1 INSECTICIDES; MITICIDES BAYER AKTIENGESELLSCHAFT (DE) 2001-01-09 US disclosed
US-5830826-A Alkoxy-alkyl-substituted 1H-3-aryl-pyrrolidine-2, 4-diones used as herbicicides and pesticides BAYER AKTIENGESELLSCHAFT (DE) 1998-11-03 US disclosed
WO-1995026954-A1 ALKOXY-ALKYL-SUBSTITUTED 1-H-3-ARYL-PYRROLIDINE-2,4-DIONES USED AS HERBICIDES AND PESTICIDES BAYER AKTIENGESELLSCHAFT (DE) 1995-10-12 WO disclosed