SCHEMBL6997866

SCHEMBL6997866

Cn1cccc1C(=O)NCCC(=O)OCc1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.66
NPC1 O15118 4/20 0.66
HRH4 Q9H3N8 1/20 0.49
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C19 P33261 1/20 0.44
PRSS1 P07477 1/20 0.44
PRSS2 P07478 1/20 0.44
ELANE P08246 1/20 0.44
PRSS3 P35030 1/20 0.44
TPSAB1 Q15661 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6991219 0.85 HRH4 (0.47) RAB9ANPC1HRH4CYP1A2CYP3A4
SCHEMBL6990088 0.84 NPC1 (0.57) RAB9ANPC1HDAC3HDAC4HDAC1
SCHEMBL6991981 0.84 CNR2 (0.56) RAB9ANPC1HRH4CYP1A2CYP3A4
SCHEMBL6654443 0.79 HRH4 (0.48) RAB9AHRH4CYP1A2CYP3A4CYP2C19
SCHEMBL12913502 0.78 PRSS1 (0.64) RAB9ANPC1HDAC2HDAC8HDAC6
SCHEMBL27441071 0.78 PRSS1 (0.69) RAB9ANPC1HRH4CYP1A2CYP3A4
SCHEMBL24526798 0.77 ALDH1A1 (0.56) HRH4CYP1A2CYP3A4CYP2C19PRSS1
SCHEMBL20201248 0.77 NPC1 (0.72) RAB9ANPC1KMT2AGAAALDH1A1
SCHEMBL13272883 0.77 NPC1 (0.73) RAB9ANPC1HDAC3HDAC4HDAC1
SCHEMBL6988747 0.76 CNR2 (0.55) RAB9ANPC1CYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0557526-B1 PYRROLOAZEPINE COMPOUND SUNTORY LTD (JP) 2003-04-02 EP disclosed
US-5399557-A Cardiovascular disorders SUNTORY LIMITED (JP) 1995-03-21 US disclosed
EP-0557526-A1 PYRROLOAZEPINE COMPOUND SUNTORY LIMITED (JP) 1993-09-01 EP disclosed