SCHEMBL6991981

SCHEMBL6991981

O=C(CCNC(=O)c1cccn1Cc1ccccc1)OCc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 6/20 0.56
HRH4 Q9H3N8 1/20 0.48
RAB9A P51151 2/20 0.45
NPC1 O15118 1/20 0.45
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C19 P33261 1/20 0.44
PRSS1 P07477 2/20 0.43
PRSS2 P07478 1/20 0.43
ELANE P08246 1/20 0.43
PRSS3 P35030 1/20 0.43
TPSAB1 Q15661 1/20 0.43
TPSD1 Q9BZJ3 1/20 0.43
TPSG1 Q9NRR2 1/20 0.43
SCN3A Q9NY46 1/20 0.43
BRD4 O60885 2/20 0.43
CNR1 P21554 2/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPK1 P28482 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6991219 0.89 HRH4 (0.47) CNR2HRH4RAB9ANPC1CYP1A2
SCHEMBL6988747 0.89 CNR2 (0.55) CNR2RAB9ANPC1CYP1A2CYP3A4
SCHEMBL6992210 0.84 CNR2 (0.64) CNR2RAB9ANPC1SCN3ABRD4
SCHEMBL6997866 0.84 RAB9A (0.66) HRH4RAB9ANPC1CYP1A2CYP3A4
SCHEMBL29020281 0.77 TDP1 (0.53) CNR2RAB9ANPC1BRD4ALDH1A1
SCHEMBL12913502 0.77 PRSS1 (0.64) RAB9ANPC1CYP1A2CYP3A4CYP2C19
SCHEMBL27441071 0.77 PRSS1 (0.69) HRH4RAB9ANPC1CYP1A2CYP3A4
SCHEMBL15576223 0.74 PRSS1 (0.59) HRH4RAB9ACYP1A2CYP3A4CYP2C19
SCHEMBL6654443 0.73 HRH4 (0.48) HRH4RAB9ACYP1A2CYP3A4CYP2C19
SCHEMBL24526798 0.73 ALDH1A1 (0.56) HRH4CYP1A2CYP3A4CYP2C19PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0557526-B1 PYRROLOAZEPINE COMPOUND SUNTORY LTD (JP) 2003-04-02 EP disclosed
US-5399557-A Cardiovascular disorders SUNTORY LIMITED (JP) 1995-03-21 US disclosed
EP-0557526-A1 PYRROLOAZEPINE COMPOUND SUNTORY LIMITED (JP) 1993-09-01 EP disclosed