SCHEMBL6998612

SCHEMBL6998612

CCOC(OCC)C1CCc2c(C(=O)O)sc(SC)c2C1=O

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.50
ALDH1A1 P00352 1/20 0.50
POLB P06746 1/20 0.50
RXFP1 Q9HBX9 1/20 0.50
NPSR1 Q6W5P4 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
CCNC P24863 4/20 0.41
CDK8 P49336 4/20 0.41
CDK19 Q9BWU1 4/20 0.41
ADORA3 P0DMS8 1/20 0.38
GAA P10253 1/20 0.35
HTT P42858 1/20 0.35
LMNA P02545 1/20 0.34
ADORA2A P29274 1/20 0.32
CDK9 P50750 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7041807 0.89 NPSR1 (0.60) KDM4EALDH1A1POLBRXFP1NPSR1
SCHEMBL7246718 0.77 MEN1 (0.46) KDM4EALDH1A1NPSR1MEN1KMT2A
SCHEMBL7248984 0.74 NPSR1 (0.44) KDM4EALDH1A1NPSR1MEN1KMT2A
SCHEMBL6987780 0.71 NPSR1 (0.63) KDM4EALDH1A1POLBRXFP1NPSR1
SCHEMBL7041221 0.68 ADORA2A (0.42) KDM4EALDH1A1NPSR1MEN1KMT2A
SCHEMBL7243172 0.68 ALDH1A1 (0.40) KDM4EALDH1A1NPSR1MEN1KMT2A
SCHEMBL6996404 0.68 NPSR1 (0.58) KDM4EALDH1A1POLBRXFP1NPSR1
SCHEMBL12663163 0.64 ALDH1A1 (0.48) KDM4EALDH1A1POLBRXFP1MEN1
SCHEMBL6988781 0.62 KDM4E (0.49) KDM4EALDH1A1POLBRXFP1NPSR1
SCHEMBL1857463 0.62 NPSR1 (1.00) KDM4EALDH1A1POLBRXFP1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268486-A2 FUSED HETEROCYCLIC DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 2003-01-02 EP disclosed
WO-2001074823-A2 FUSED HETEROCYCLIC DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-10-11 WO disclosed