SCHEMBL6999520

SCHEMBL6999520

O=CN1CCC(C(=O)c2ccc(Cl)cc2)CC1

nearest known ligand 0.65

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 14/20 0.65
MEN1 O00255 1/20 0.62
KMT2A Q03164 1/20 0.62
LMNA P02545 1/20 0.58
TP53 P04637 1/20 0.58
MAPT P10636 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
HSD11B1 P28845 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8105526 0.91 MGLL (0.58) MGLLMEN1KMT2ALMNATP53
SCHEMBL4500344 0.85 HTR2A (0.56) MGLLMEN1KMT2ALMNAHSD11B1
SCHEMBL27892705 0.84 KMT2A (0.65) MGLLMEN1KMT2ALMNAHSD11B1
SCHEMBL4509082 0.84 HSD11B1 (0.65) MGLLHSD11B1
SCHEMBL13657578 0.81 MGLL (0.71) MGLLMEN1KMT2ALMNATP53
SCHEMBL28975834 0.81 POLB (0.57) MGLLMEN1KMT2AHSD11B1
(4-Chlorophenyl)(Cyclopropyl)Methanone SCHEMBL392801 0.80 MGLL (0.68) MGLLMEN1KMT2ALMNATP53
SCHEMBL14154609 0.80 MGLL (0.69) MGLLMEN1KMT2ALMNATP53
SCHEMBL3391998 0.80 MGLL (0.69) MGLLMEN1KMT2ALMNATP53
SCHEMBL10638259 0.79 MGLL (0.45) MGLLMEN1KMT2AHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6670379-B2 Inflammatory or allergic conditions, asthma, inhibition of eosinophil activation, conjunctivitis; (1-((R2-Amino-3-pyridin-3-yl-propyl)-piperidin-4-yl)-(4-fluoro-phenyl) -methanone NOVARTIS AG (CH) 2003-12-30 US disclosed
US-20030176460-A1 Piperidine compounds for use as ccr-3 inhibitors NOVARTIS AG (CH) 2003-09-18 US disclosed
EP-1303488-A1 PIPERIDINE COMPOUNDS FOR USE AS CCR-3 INHIBITORS Novartis AG (CH) 2003-04-23 EP disclosed
WO-2002004420-A1 PIPERIDINE COUMPOUNDS FOR USE AS CCR-3 INHIBITORS NOVARTIS AG (CH) 2002-01-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030176460-A1 Piperidine compounds for use as ccr-3 inhibitors CCR1, CCR3, CCR4 MGLL 4087/4885MEN1 4248/4885KMT2A 3218/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.