SCHEMBL7000554

SCHEMBL7000554

Nc1nc2c(c(=O)[nH]1)S[C@@H](CCc1ccc(C(=O)O)s1)CN2

nearest known ligand 0.71

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GART P22102 8/20 0.71
FOLR1 P15328 11/20 0.53
NOS1 P29475 1/20 0.38
FOLR2 P14207 3/20 0.38
DHFR P00374 1/20 0.36
SLC46A1 Q96NT5 3/20 0.35
ATIC P31939 2/20 0.35
SLC19A1 P41440 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6996555 1.00 GART (0.71) GARTFOLR1NOS1FOLR2DHFR
SCHEMBL22967335 0.85 GART (0.59) GARTFOLR1NOS1ATIC
SCHEMBL10067962 0.84 GART (1.00) GARTFOLR1FOLR2SLC46A1ATIC
SCHEMBL24846050 0.82 GART (0.57) GARTFOLR1NOS1DHFRATIC
SCHEMBL7812453 0.82 GART (0.69) GARTFOLR1NOS1ATIC
SCHEMBL6991867 0.82 GART (0.72) GARTFOLR1NOS1ATIC
SCHEMBL6993317 0.82 GART (0.72) GARTFOLR1NOS1ATIC
SCHEMBL8362067 0.74 GART (0.53) GARTFOLR1NOS1ATIC
SCHEMBL6996839 0.73 GART (0.66) GARTFOLR1NOS1ATIC
SCHEMBL7825368 0.70 GART (1.00) GARTFOLR1ATIC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0846111-B1 SYNTHESES OF OPTICALLY PURE COMPOUNDS USEFUL AS GARFT INHIBITORS AND THEIR INTERMEDIATES AGOURON PHARMA (US) 2003-08-27 EP disclosed
US-5981748-A Synthesis of optically pure compounds useful as GARFT inhibitors and their intermediates AGOURON PHARMACEUTICALS, INC. (US) 1999-11-09 US disclosed