SCHEMBL6993317

SCHEMBL6993317

Cc1cc(C(=O)O)sc1CC[C@H]1CNc2nc(N)[nH]c(=O)c2S1

nearest known ligand 0.72

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GART P22102 7/20 0.72
FOLR1 P15328 4/20 0.72
NOS1 P29475 6/20 0.34
NOS3 P29474 1/20 0.34
NOS2 P35228 1/20 0.34
ATIC P31939 2/20 0.33
USP2 O75604 1/20 0.32
CASP7 P55210 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6991867 1.00 GART (0.72) GARTFOLR1NOS1NOS3NOS2
SCHEMBL6996839 0.89 GART (0.66) GARTFOLR1NOS1NOS3NOS2
SCHEMBL7000554 0.82 GART (0.71) GARTFOLR1NOS1ATIC
SCHEMBL7145433 0.80 GART (0.80) GARTFOLR1ATIC
SCHEMBL8362067 0.79 GART (0.53) GARTFOLR1NOS1NOS3NOS2
SCHEMBL7812453 0.77 GART (0.69) GARTFOLR1NOS1ATIC
SCHEMBL8537889 0.77 GART (0.63) GARTFOLR1ATIC
SCHEMBL22967335 0.76 GART (0.59) GARTFOLR1NOS1NOS3NOS2
SCHEMBL24846050 0.72 GART (0.57) GARTFOLR1NOS1NOS3NOS2
Pelitrexol SCHEMBL13916067 0.68 GART (0.74) GARTFOLR1ATIC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0846111-B1 SYNTHESES OF OPTICALLY PURE COMPOUNDS USEFUL AS GARFT INHIBITORS AND THEIR INTERMEDIATES AGOURON PHARMA (US) 2003-08-27 EP disclosed
US-5981748-A Synthesis of optically pure compounds useful as GARFT inhibitors and their intermediates AGOURON PHARMACEUTICALS, INC. (US) 1999-11-09 US disclosed