SCHEMBL7001602

SCHEMBL7001602

CC(C)(C)OC(=O)Nc1ccccc1CCc1nc(-c2ccccc2)no1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
HDAC1 Q13547 3/20 0.48
HDAC2 Q92769 3/20 0.48
HPGD P15428 2/20 0.48
CYP1A2 P05177 2/20 0.48
CYP2C19 P33261 2/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
TSHR P16473 3/20 0.47
LMNA P02545 2/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 3/20 0.47
MAPK1 P28482 2/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
HCAR2 Q8TDS4 1/20 0.47
HTT P42858 1/20 0.47
HDAC8 Q9BY41 2/20 0.47
CYP2D6 P10635 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14846086 0.82 CYP1A2 (0.58) ALDH1A1HDAC1HDAC2HPGDCYP1A2
SCHEMBL29096990 0.78 ALDH1A1 (0.50) ALDH1A1HDAC1HDAC2HPGDCYP1A2
SCHEMBL14736015 0.77 PDE10A (0.52) ALDH1A1HPGDNPC1RAB9ATSHR
SCHEMBL29828943 0.77 HPGD (0.49) ALDH1A1HDAC1HDAC2HPGDCYP1A2
SCHEMBL6323275 0.76 HTT (0.57) ALDH1A1HDAC1HDAC2HPGDTSHR
SCHEMBL1610079 0.76 TSHR (0.51) ALDH1A1HPGDCYP1A2CYP2C19TSHR
SCHEMBL6802648 0.75 LMNA (0.45) LMNA
SCHEMBL1772002 0.74 LMNA (0.47) ALDH1A1TSHRLMNA
SCHEMBL5757395 0.74 POLB (0.47) ALDH1A1TSHRLMNA
SCHEMBL12474847 0.74 POLB (0.42) NPC1RAB9ALMNAMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317459-A1 BICYCLIC PYRROLYL AMIDES AS GLUCOGEN PHOSPHORYLASE INHIBITORS AstraZeneca AB (SE) 2003-06-11 EP disclosed
WO-2002020530-A1 BICYCLIC PYRROLYL AMIDES AS GLUCOGEN PHOSPHORYLASE INHIBITORS ASTRAZENECA AB (SE) 2002-03-14 WO disclosed