SCHEMBL7001776

SCHEMBL7001776

CC1=C(N)Nc2cc(C(C)(N)c3cccs3)ccc2O1

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ACE2 Q9BYF1 1/20 0.35
ESR1 P03372 1/20 0.32
CNR1 P21554 2/20 0.30
CNR2 P34972 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6988641 0.99 ACE2 (0.34) ACE2ESR1CNR1CNR2
Hydrochloric Acid SCHEMBL6992620 0.85 ACE2 (0.32) ACE2ESR1
Hydrochloric Acid SCHEMBL6999219 0.83 ESR1 (0.33) ACE2ESR1
Hydrochloric Acid SCHEMBL8119304 0.82 GAA (0.35)
Hydrochloric Acid SCHEMBL8118427 0.81 ESR1 (0.31) ESR1
SCHEMBL7988325 0.80 ALDH1A1 (0.36) ACE2
SCHEMBL6996954 0.80 ACE2 (0.32) ACE2
Hydrochloric Acid SCHEMBL6991848 0.79 ACE2 (0.31) ACE2
SCHEMBL7708334 0.78 ALDH1A1 (0.32) ACE2
SCHEMBL7003121 0.76 KCNH2 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015437-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AG (DE) 2003-12-03 EP claimed