SCHEMBL7708334

SCHEMBL7708334

CC1=C(N)Nc2cc(C(C)(NC(=O)OC(C)(C)C)c3cccs3)ccc2O1

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.32
MAPK10 P53779 1/20 0.31
POLB P06746 1/20 0.31
GAA P10253 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CTSS P25774 1/20 0.31
CTSK P43235 1/20 0.31
ACE2 Q9BYF1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7704890 0.89 CTSK (0.32) CTSSCTSK
SCHEMBL7710991 0.88 CTSK (0.32) ALDH1A1CTSSCTSK
SCHEMBL7710849 0.85 MAPK10 (0.31) MAPK10ACE2
SCHEMBL7708011 0.83 LATS1 (0.34) MAPK10
SCHEMBL7711551 0.83 NPC1 (0.33) MAPK10SMN1; SMN2
SCHEMBL7711067 0.81 NAMPT (0.36) ALDH1A1
SCHEMBL7705086 0.81 NPSR1 (0.35) MAPK10GAA
SCHEMBL7711428 0.80 PARP1 (0.39) ALDH1A1MAPK10GAA
SCHEMBL7089637 0.80 ALDH1A1 (0.32) ALDH1A1MAPK10
SCHEMBL7713259 0.78 USP2 (0.39) ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed