SCHEMBL700206

SCHEMBL700206

O=C(O)[C@@H]1C[C@@H](S(=O)(=O)c2ccc(N3CCCCC3)cc2Cl)CN1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSS P25774 11/20 0.45
CTSL P07711 4/20 0.40
CTSB P07858 4/20 0.40
CTSK P43235 2/20 0.40
NOTUM Q6P988 1/20 0.40
HSD11B1 P28845 3/20 0.40
LMNA P02545 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
GFER P55789 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3065886 0.92 CTSS (0.46) CTSSCTSLCTSBCTSKNOTUM
SCHEMBL3807046 0.85 CTSS (0.40) CTSSCTSLCTSBCTSKNOTUM
SCHEMBL3060577 0.85 CTSS (0.40) CTSSCTSLCTSBCTSKNOTUM
SCHEMBL3073598 0.85 CTSS (0.58) CTSS
SCHEMBL700379 0.84 CTSS (0.67) CTSSCTSLCTSB
SCHEMBL3065798 0.81 CTSL (0.59) CTSSCTSLCTSBCTSK
SCHEMBL698949 0.80 CTSS (0.46) CTSSCTSLCTSB
SCHEMBL3073773 0.78 DPP4 (0.40) CTSSNOTUMHSD11B1LMNAMEN1
Lithium Ion SCHEMBL2106607 0.78 CTSS (0.42) CTSSCTSLCTSBCTSKHSD11B1
SCHEMBL2102652 0.78 NR1H2 (0.47) CTSSCTSLCTSBCTSKHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP disclosed
WO-2010121918-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-10-28 WO disclosed