SCHEMBL7002285

SCHEMBL7002285

CCCCOc1c2cc(=O)c(F)cc-2cn(CC(C)(C)C)c1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.38
RARB P10826 5/20 0.36
RARA P10276 3/20 0.36
FFAR4 Q5NUL3 6/20 0.33
FFAR1 O14842 3/20 0.33
PLA2G2A P14555 1/20 0.33
THRA P10827 1/20 0.32
THRB P10828 1/20 0.32
RARG P13631 2/20 0.32
GRIN2D O15399 1/20 0.31
GRIN3B O60391 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2A Q12879 1/20 0.31
GRIN2B Q13224 1/20 0.31
GRIN2C Q14957 1/20 0.31
GRIN3A Q8TCU5 1/20 0.31
PPARD Q03181 1/20 0.31
CNR2 P34972 1/20 0.30
PTPN11 Q06124 1/20 0.30
NR4A2 P43354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7555530 0.84 MCL1 (0.38) MCL1RARBRARATHRATHRB
SCHEMBL7006171 0.79 ESR1 (0.34) FFAR4THRATHRBCNR2
SCHEMBL7003231 0.75 SLC6A5 (0.38) CNR2
SCHEMBL7007505 0.74 SLC6A5 (0.37) CNR2
SCHEMBL7006105 0.73 SLC6A5 (0.33) MCL1THRATHRB
SCHEMBL7007513 0.73 THRA (0.32) FFAR4THRATHRB
SCHEMBL7001088 0.73 NPC1 (0.36) MCL1RARB
SCHEMBL7559138 0.73 FFAR4 (0.35) FFAR4
SCHEMBL7004588 0.72 SLC6A5 (0.38) FFAR4CNR2
SCHEMBL7004682 0.72 SLC6A5 (0.32) FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355886-A1 FUSED HETEROCYCLIC COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2003-10-29 EP disclosed
WO-2002062764-A9 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-10-10 WO disclosed
WO-2002062764-A1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-08-15 WO disclosed