SCHEMBL7002876

SCHEMBL7002876

CCOCc1ccc2nc3ccc(=O)cc-3oc2c1

nearest known ligand 0.66

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
APP P05067 13/20 0.66
CYP1A2 P05177 1/20 0.66
MEN1 O00255 2/20 0.33
POLB P06746 2/20 0.33
RAB9A P51151 2/20 0.33
KMT2A Q03164 2/20 0.33
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
ALPL P05186 1/20 0.33
ALPI P09923 1/20 0.33
ALPG P10696 1/20 0.33
RECQL P46063 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
NPC1 O15118 2/20 0.32
TP53 P04637 1/20 0.31
TRPV1 Q8NER1 1/20 0.31
SNCA P37840 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6998321 0.87 APP (0.67) APPCYP1A2MEN1POLBRAB9A
SCHEMBL1093926 0.86 APP (0.60) APPCYP1A2MEN1POLBRAB9A
SCHEMBL119047 0.86 APP (0.56) APPCYP1A2KMT2AMAPTALDH1A1
SCHEMBL563769 0.85 APP (0.66) APPCYP1A2MEN1POLBRAB9A
Ether SCHEMBL1094032 0.85 APP (0.80) APPCYP1A2MEN1POLBKMT2A
SCHEMBL1104922 0.81 APP (0.82) APPCYP1A2
SCHEMBL10167845 0.80 APP (0.68) APPCYP1A2MEN1POLBRAB9A
SCHEMBL738742 0.80 APP (0.59) APPCYP1A2MAPT
Ethoxyresorufin SCHEMBL104497 0.80 APP (1.00) APPCYP1A2
Ethoxyresorufin SCHEMBL31079400 0.80 APP (1.00) APPCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140888-B1 OPTICAL MOLECULAR SENSORS FOR CYTOCHROME P450 ACTIVITY VERTEX PHARMA SAN DIEGO LLC (US) 2003-05-14 EP claimed
US-6420130-B1 CHEMICAL COMPOUND FOR USE IN THE DETECTION OF PREFERENTIAL ENZYMATIC POLYPEPTIDE AURORA BIOSCIENCES CORPORATION 2002-07-16 US claimed