SCHEMBL7002987

SCHEMBL7002987

C[C@H]1CCCCN1C(=O)OC(C)(C)C

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.49
GAA P10253 1/20 0.49
HSD17B10 Q99714 1/20 0.48
EPHX1 P07099 1/20 0.45
PREP P48147 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7005690 1.00 HPGD (0.49) HPGDGAAHSD17B10EPHX1PREP
SCHEMBL1202111 1.00 HPGD (0.49) HPGDGAAHSD17B10EPHX1PREP
SCHEMBL357043 0.95 HSD17B10 (0.52) HPGDHSD17B10EPHX1SMN1; SMN2NPC1
SCHEMBL178721 0.95 HSD17B10 (0.52) HPGDHSD17B10EPHX1SMN1; SMN2NPC1
SCHEMBL357042 0.95 HSD17B10 (0.52) HPGDHSD17B10EPHX1SMN1; SMN2NPC1
SCHEMBL31539240 0.88 HPGD (0.48) HPGDHSD17B10EPHX1PREPSMN1; SMN2
SCHEMBL27618621 0.88 PREP (0.42) HPGDGAAHSD17B10EPHX1PREP
SCHEMBL4175218 0.87 CHRM2 (0.44) HPGDHSD17B10EPHX1PREPSMN1; SMN2
SCHEMBL489128 0.87 CHRM2 (0.44) HPGDHSD17B10EPHX1PREPSMN1; SMN2
SCHEMBL489126 0.87 CHRM2 (0.44) HPGDHSD17B10EPHX1PREPSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250206724-A1 SUBSTITUTED 3-AMINO INDAZOLE DERIVATIVES AS KINASE INHIBITORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2025-06-26 US disclosed
EP-4499612-A1 SUBSTITUTED 3-AMINO INDAZOLE DERIVATIVES AS KINASE INHIBITORS Nerviano Medical Sciences S.r.l. (IT) 2025-02-05 EP disclosed
CN-118974020-A Substituted 3-aminoindazole derivatives as kinase inhibitors 内尔维亚诺医疗科学公司 2024-11-15 CN disclosed
WO-2023186773-A1 SUBSTITUTED 3-AMINO INDAZOLE DERIVATIVES AS KINASE INHIBITORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2023-10-05 WO disclosed
US-11766436-B2 KRAS G12C inhibitors and methods of using the same AMGEN INC. (US) 2023-09-26 US disclosed
EP-4198024-A1 PYRAZOLE MAGL INHIBITORS H. Lundbeck A/S (DK) 2023-06-21 EP disclosed
US-20210309638-A1 3-(1-OXOISOINDOLIN-2-YL)PIPERIDINE-2,6-DIONE DERIVATIVES AND USES THEREOF NOVARTIS AG (CH) 2021-10-07 US disclosed
US-11053218-B2 3-(1-oxoisoindolin-2-yl)piperidine-2,6-dione derivatives and uses thereof NOVARTIS AG (CH) 2021-07-06 US disclosed
US-20200231569-A1 3-(1-OXOISOINDOLIN-2-YL)PIPERIDINE-2,6-DIONE DERIVATIVES AND USES THEREOF NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2020-07-23 US disclosed
WO-2020028115-A1 5-METHYL-4-FLUORO-THIAZOL-2-YL COMPOUNDS ELI LILLY AND COMPANY (US) 2020-02-06 WO disclosed
US-8987250-B2 Therapeutic compounds GILEAD SCIENCES, INC. (US) 2015-03-24 US disclosed
US-20140343042-A1 NICOTINE RECEPTOR TARGETED COMPOUNDS AND COMPOSITIONS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. 2014-11-20 US disclosed
US-20130281433-A1 THERAPEUTIC COMPOUNDS GILEAD SCIENCES, INC. 2013-10-24 US disclosed
US-8461328-B2 Tricyclic heterocyclic compounds, compositions and methods of use thereof GENENTECH, INC. (US) 2013-06-11 US disclosed
US-8461328-B2 Tricyclic heterocyclic compounds, compositions and methods of use thereof GENENTECH, INC. (US) 2013-06-11 US disclosed
US-20110201593-A1 TRICYCLIC HETEROCYCLIC COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2011-08-18 US disclosed
CN-1863797-A Cyclic amine BACE-1 inhibitors having a benzamide substituent PHARMACOPEIA DRUG DISCOVERY (US) 2006-11-15 CN disclosed
EP-1138679-B1 HYDRONAPHTHO 2,3-c]FURAN DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF SAGAMI CHEM RES (JP) 2003-03-19 EP disclosed
US-6392059-B1 THERAPY FOR ALZHEIMER'S DISEASE SAGAMI CHEMICAL REASEARCH CENTER (JP) 2002-05-21 US disclosed
EP-1138679-A1 HYDRONAPHTHO 2,3-c]FURAN DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF SAGAMI CHEMICAL RESEARCH CENTER (JP) 2001-10-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250206724-A1 SUBSTITUTED 3-AMINO INDAZOLE DERIVATIVES AS KINASE INHIBITORS CDK1, CDK11A, CDK3 HPGD 2141/4885GAA 3479/4885HSD17B10 3713/4885
US-20130281433-A1 THERAPEUTIC COMPOUNDS NQO1, HAVCR2, CCR5 HPGD 656/4885GAA 42/4885HSD17B10 1005/4885
US-20210309638-A1 3-(1-OXOISOINDOLIN-2-YL)PIPERIDINE-2,6-DIONE DERIVATIVES AND USES THEREOF XDH, H1-0, RXFP1 HPGD 888/4885GAA 1642/4885HSD17B10 3610/4885
US-20110201593-A1 TRICYCLIC HETEROCYCLIC COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF CCNY, CCNA1, CCNA2 HPGD 223/4885GAA 2545/4885HSD17B10 863/4885
US-20140343042-A1 NICOTINE RECEPTOR TARGETED COMPOUNDS AND COMPOSITIONS CHRNA7, CHRNA5, CHRNA4 HPGD 2162/4885GAA 1933/4885HSD17B10 1854/4885
US-20200231569-A1 3-(1-OXOISOINDOLIN-2-YL)PIPERIDINE-2,6-DIONE DERIVATIVES AND USES THEREOF XDH, H1-0, RXFP1 HPGD 888/4885GAA 1642/4885HSD17B10 3610/4885
US-11766436-B2 KRAS G12C inhibitors and methods of using the same KRAS, NRAS, HRAS HPGD 2130/4885GAA 2321/4885HSD17B10 3826/4885
US-11053218-B2 3-(1-oxoisoindolin-2-yl)piperidine-2,6-dione derivatives and uses thereof XDH, H1-0, RXFP1 HPGD 888/4885GAA 1642/4885HSD17B10 3610/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.