SCHEMBL7003015

SCHEMBL7003015

CC(C)(C)[Si](C)(C)OCCCc1cccc(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 5/20 0.44
CYP3A4 P08684 2/20 0.42
IDO1 P14902 2/20 0.42
AGXT P21549 2/20 0.42
AOC3 Q16853 1/20 0.42
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
HTR3A P46098 1/20 0.42
HTR3D Q70Z44 1/20 0.42
HTR3C Q8WXA8 1/20 0.42
MAOB P27338 1/20 0.40
PNMT P11086 2/20 0.39
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15413373 0.91 TAAR1 (0.46) TAAR1CYP3A4IDO1AGXTAOC3
SCHEMBL19438938 0.87 CHRM2 (0.47) TAAR1CHRM2
SCHEMBL21268599 0.82 IDO1 (0.42) IDO1
SCHEMBL3168839 0.82 GABRA1 (0.47) TAAR1CHRM2CHRM1CHRM3
SCHEMBL21068770 0.82 DUT (0.37) IDO1
SCHEMBL11482682 0.82 DUT (0.37) IDO1CHRM2CHRM1CHRM3
SCHEMBL3643273 0.82 TAAR1 (0.44) TAAR1IDO1AGXTMAOB
SCHEMBL21367138 0.81 CYP3A4 (0.56) TAAR1CYP3A4IDO1AGXTMAOB
SCHEMBL30859481 0.81 DUT (0.40) TAAR1CYP3A4IDO1AGXTAOC3
SCHEMBL2252126 0.81 IDO1 (0.53) IDO1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1325011-A2 METHODS AND COMPOUNDS FOR TREATING PROLIFERATIVE DISEASES ELI LILLY AND COMPANY (US) 2003-07-09 EP disclosed
WO-2002028861-A2 METHODS AND COMPOUNDS FOR TREATING PROLIFERATIVE DISEASES ELI LILLY AND COMPANY (US) 2002-04-11 WO disclosed