SCHEMBL7003228

SCHEMBL7003228

CC(C)(C)c1cc(OCc2nccn2Cc2ccccc2)nn2c(-c3cc(Cl)on3)nnc12

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 12/20 0.44
GABRG2 P18507 12/20 0.44
GABRB3 P28472 12/20 0.44
GABRA3 P34903 12/20 0.44
GABRA5 P31644 11/20 0.44
GABRA2 P47869 11/20 0.44
GABRA4 P48169 1/20 0.36
GABRA6 Q16445 1/20 0.36
HSP90AA1 P07900 2/20 0.35
CACNA2D1 P54289 1/20 0.34
ERBB2 P04626 1/20 0.34
EPHA2 P29317 1/20 0.34
KDR P35968 1/20 0.34
EPHB4 P54760 1/20 0.34
PDE5A O76074 2/20 0.33
HSP90AB1 P08238 1/20 0.33
HSP90B1 P14625 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7001121 0.92 GABRA1 (0.44) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL7003553 0.90 GABRA1 (0.44) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL7003230 0.83 GABRA1 (0.49) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL6998714 0.79 GABRG2 (0.48) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL2657628 0.76 GABRA1 (0.50) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL7003676 0.76 GABRA1 (0.51) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL7003973 0.75 GABRA1 (0.52) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL7487491 0.74 GABRA1 (0.67) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL6999458 0.73 GABRA1 (0.66) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL7003556 0.73 GABRA1 (0.47) GABRA1GABRG2GABRB3GABRA3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1107967-B1 TRIAZOLOPYRIDAZINE DERIVATIVES FOR ENHANCING COGNITION MERCK SHARP & DOHME (GB) 2003-05-14 EP claimed