SCHEMBL7003543

SCHEMBL7003543

CC(C)Cn1c(C(=O)O)c(OS(=O)(=O)C(F)(F)F)c2ccccc2c1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.49
TSHR P16473 2/20 0.49
HSD17B10 Q99714 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
DPP4 P27487 6/20 0.41
ALDH1A1 P00352 6/20 0.40
KDM4E B2RXH2 4/20 0.39
KMT2A Q03164 4/20 0.38
MEN1 O00255 3/20 0.38
LMNA P02545 2/20 0.37
USP2 O75604 1/20 0.37
GAA P10253 1/20 0.37
HTT P42858 1/20 0.37
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
PER2 O15055 1/20 0.37
CRY1 Q16526 1/20 0.37
CRY2 Q49AN0 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5234705 0.76 MAPK8 (0.44) DPP4
SCHEMBL5237348 0.75 DPP4 (0.40) DPP4
SCHEMBL12499481 0.74 ALDH1A1 (0.43) SMN1; SMN2HSD17B10ALDH1A1KDM4EKMT2A
SCHEMBL5577125 0.70 CCR2 (0.33) DPP4GAAPOLB
SCHEMBL12687183 0.69 EGFR (0.41) SMN1; SMN2TSHRHSD17B10L3MBTL1ALDH1A1
SCHEMBL5233740 0.68 DPP4 (0.49) DPP4
SCHEMBL4713112 0.68 MAPK8 (0.59) PTGS1PTGS2
SCHEMBL15093426 0.66 CXCR2 (0.34) SMN1; SMN2HSD17B10LMNAHTTPER2
SCHEMBL15099628 0.65 HTT (0.39) SMN1; SMN2TSHRHSD17B10ALDH1A1KDM4E
SCHEMBL5235433 0.65 DPP4 (0.69) DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355886-A1 FUSED HETEROCYCLIC COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2003-10-29 EP disclosed
WO-2002062764-A1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-08-15 WO disclosed