SCHEMBL7004388

SCHEMBL7004388

COc1ccc(Cc2ccc3nc4ccc(=O)cc-4oc3c2)cc1

nearest known ligand 0.76

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
APP P05067 13/20 0.76
CYP1A2 P05177 1/20 0.63
NPC1 O15118 4/20 0.43
RAB9A P51151 4/20 0.43
KMT2A Q03164 1/20 0.43
POLB P06746 1/20 0.41
LMNA P02545 1/20 0.41
TLR4 O00206 1/20 0.41
XDH P47989 1/20 0.41
NLRP3 Q96P20 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31115697 0.86 APP (1.00) APPCYP1A2NPC1RAB9ALMNA
SCHEMBL563392 0.86 APP (1.00) APPCYP1A2NPC1RAB9ALMNA
SCHEMBL1104921 0.86 APP (1.00) APPCYP1A2NPC1RAB9AKMT2A
SCHEMBL1094100 0.85 APP (0.59) APPCYP1A2RAB9AKMT2APOLB
SCHEMBL10167882 0.83 APP (1.00) APPCYP1A2NPC1RAB9A
SCHEMBL6998321 0.83 APP (0.67) APPCYP1A2NPC1RAB9AKMT2A
SCHEMBL563769 0.81 APP (0.66) APPCYP1A2NPC1RAB9AKMT2A
SCHEMBL10167883 0.81 APP (0.93) APPCYP1A2
SCHEMBL10167845 0.78 APP (0.68) APPCYP1A2RAB9AKMT2APOLB
SCHEMBL7002876 0.78 APP (0.66) APPCYP1A2NPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140888-B1 OPTICAL MOLECULAR SENSORS FOR CYTOCHROME P450 ACTIVITY VERTEX PHARMA SAN DIEGO LLC (US) 2003-05-14 EP claimed
US-6143492-A COMPOUND USEFUL AS AN OPTICAL PROBE; DRUG SCREENING AURORA BIOSCIENCES CORPORATION (US) 2000-11-07 US claimed