SCHEMBL7005559

SCHEMBL7005559

Cn1cc2c(=O)c(Cl)c(Cl)cc-2c(-c2ccccc2)c1C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.42
BRD4 O60885 2/20 0.37
KDM4E B2RXH2 2/20 0.36
GRIA4 P48058 5/20 0.36
GRIA2 P42262 4/20 0.36
MEN1 O00255 2/20 0.35
RAB9A P51151 1/20 0.35
PKM P14618 1/20 0.34
HKDC1 Q2TB90 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CYP2C9 P11712 1/20 0.34
CREBBP Q92793 1/20 0.34
FABP3 P05413 1/20 0.34
FABP4 P15090 1/20 0.34
ACLY P53396 1/20 0.34
HSP90AA1 P07900 1/20 0.33
TTR P02766 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7008527 0.85 BAZ2B (0.45) KMT2AKDM4EMEN1RAB9ACYP2C9
SCHEMBL7555153 0.79 BRD4 (0.36) KMT2ABRD4KDM4EGRIA4GRIA2
SCHEMBL1081579 0.70 GRIA4 (0.47) KMT2ABRD4KDM4EGRIA4GRIA2
SCHEMBL1381646 0.69 HK2 (0.40) BRD4GRIA4GRIA2CREBBPFABP3
SCHEMBL1254367 0.67 BRD4 (0.47) KMT2ABRD4KDM4EGRIA4GRIA2
SCHEMBL8287396 0.66 GRIA4 (0.59) GRIA4GRIA2
SCHEMBL5231452 0.66 DPP4 (0.46) GRIA4GRIA2
SCHEMBL31154485 0.64 CYP2C9 (0.37) KMT2AKDM4EMEN1PKMCYP2C9
SCHEMBL2637715 0.64 GRIA2 (0.45) KDM4EGRIA4GRIA2RAB9A
SCHEMBL8289845 0.64 GRIA4 (0.57) KDM4EGRIA4GRIA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355886-A1 FUSED HETEROCYCLIC COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2003-10-29 EP disclosed
WO-2002062764-A1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-08-15 WO disclosed