SCHEMBL7005697

SCHEMBL7005697

O=C(C1CCCN(CCCc2ccccc2)C1)C1CCCN(CCCc2ccccc2)C1

nearest known ligand 0.75

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.75
KMT2A Q03164 1/20 0.75
GAA P10253 1/20 0.65
CHRNB2 P17787 5/20 0.62
CHRNB4 P30926 5/20 0.62
CHRNA3 P32297 5/20 0.62
CHRNA4 P43681 5/20 0.62
ALDH1A1 P00352 1/20 0.58
BLM P54132 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28747604 0.88 KDM4E (0.70) KDM4EKMT2A
SCHEMBL8873337 0.83 SLC6A1 (0.65)
Hydrochloric Acid SCHEMBL8871870 0.82 SLC6A1 (0.64)
SCHEMBL947855 0.82 KDM4E (0.62) KDM4EKMT2ACHRNB2CHRNB4CHRNA3
SCHEMBL10523377 0.81 KDM4E (0.61) KDM4EKMT2A
SCHEMBL10523381 0.81 ALDH1A1 (0.68) KDM4EKMT2AALDH1A1
SCHEMBL28747644 0.81 CHRNB4 (0.62) KDM4EKMT2ACHRNB2CHRNB4CHRNA3
SCHEMBL2450443 0.81 KMT2A (0.60) KDM4EKMT2AGAA
SCHEMBL3575018 0.80 KDM4E (0.60) KDM4EKMT2AGAACHRNB2CHRNB4
SCHEMBL18593785 0.79 S1PR1 (0.67) KDM4EKMT2AALDH1A1BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242080-A4 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE UNIV GEORGETOWN (US) 2003-01-22 EP claimed
EP-1242080-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2002-09-25 EP claimed
WO-2001022964-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2001-04-05 WO claimed