SCHEMBL7005836

SCHEMBL7005836

O=C(OCc1ccccc1)OC1CCCN1C(=O)c1ccncc1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.46
CYP2D6 P10635 3/20 0.46
GRIN2B Q13224 2/20 0.46
SPHK2 Q9NRA0 2/20 0.44
CYP3A4 P08684 3/20 0.44
CYP1A2 P05177 1/20 0.44
SPHK1 Q9NYA1 1/20 0.44
PREP P48147 6/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
POLB P06746 1/20 0.41
TSHR P16473 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6291342 0.82 FKBP1A (0.57) SPHK2SPHK1PREP
SCHEMBL7009968 0.81 KDM4E (0.49) PREPNPC1POLB
SCHEMBL1578423 0.77 SPHK2 (0.52) SPHK2SPHK1NPC1RAB9ASMN1; SMN2
SCHEMBL4602471 0.76 PREP (0.54) PREPNPC1RAB9ASMN1; SMN2TSHR
SCHEMBL11848922 0.74 SMN1; SMN2 (0.50) NPC1RAB9ASMN1; SMN2CYP2C19
SCHEMBL13149480 0.74 CYP2D6 (0.60) CYP2C9CYP2D6GRIN2BCYP3A4NPC1
SCHEMBL6788581 0.72 FKBP1A (0.63) SPHK2SPHK1PREP
SCHEMBL6788577 0.72 FKBP1A (0.63) SPHK2SPHK1PREP
SCHEMBL10452175 0.72 FKBP1A (0.46) GRIN2BPREPNPC1RAB9ASMN1; SMN2
SCHEMBL7284521 0.70 SMN1; SMN2 (0.54) PREPNPC1RAB9ASMN1; SMN2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1252163-B1 4-PYRIDYL-AND 2,4-PYRIMIDINYL-SUBSTITUTED PYRROLE DERIVATIVES AND THEIR USE IN PHARMACY MERCKLE GMBH (DE) 2003-09-24 EP disclosed
EP-1252163-A2 4-PYRIDYL-AND 2,4-PYRIMIDINYL-SUBSTITUTED PYRROLE DERIVATIVES AND THEIR USE IN PHARMACY MERCKLE GMBH (DE) 2002-10-30 EP disclosed
WO-2001057042-A2 4-PYRIDYL-AND 2,4-PYRIMIDINYL-SUBSTITUTED PYRROLE DERIVATIVES AND THEIR USE IN PHARMACY MERCKLE GMBH (DE) 2001-08-09 WO disclosed