SCHEMBL7007102

SCHEMBL7007102

CCOC(=O)c1cn(C2CC2)c2c(OCF)c(-c3ccc4c(c3)CN(S(=O)(=O)c3ccc(C)cc3)C4)c(F)cc2c1=O

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.42
TOP2A P11388 6/20 0.40
TOP2B Q02880 6/20 0.40
HPGD P15428 1/20 0.40
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
KMT2A Q03164 1/20 0.39
KCNH2 Q12809 2/20 0.35
GSK3B P49841 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HDAC1 Q13547 1/20 0.34
GAA P10253 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7010122 0.93 ADRB2 (0.43) ADRB2TOP2ATOP2BHPGDMEN1
SCHEMBL7014704 0.92 TOP2A (0.49) TOP2ATOP2BHPGDMEN1KMT2A
SCHEMBL7010280 0.91 ADRB2 (0.42) ADRB2TOP2ATOP2BHPGDMEN1
SCHEMBL7008688 0.91 ADRB2 (0.45) ADRB2TOP2ATOP2BHPGDMEN1
SCHEMBL7010320 0.91 TOP2A (0.49) ADRB2TOP2ATOP2BHPGDMEN1
SCHEMBL7008129 0.90 ADRB2 (0.44) ADRB2TOP2ATOP2BHPGDMEN1
SCHEMBL7007624 0.84 TOP2A (0.49) TOP2ATOP2BHPGDMEN1KMT2A
SCHEMBL7509004 0.83 ADRB2 (0.44) ADRB2TOP2ATOP2BHPGDMEN1
SCHEMBL7010716 0.83 HPGD (0.45) ADRB2HPGDMEN1MAPTTHRB
SCHEMBL8323507 0.82 KMT2A (0.42) ADRB2HPGDMEN1MAPTTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775702-B1 NOVEL QUINOLONE- OR NAPHTHYRIDONECARBOXYLIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO LTD (JP) 2003-07-23 EP disclosed
US-5935952-A ANTIBACTERIAL AGENT TOYAMA CHEMICAL CO., LTD. (JP) 1999-08-10 US disclosed
EP-0775702-A1 NOVEL QUINOLONE- OR NAPHTHYRIDONECARBOXYLIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 1997-05-28 EP disclosed