SCHEMBL7007499

SCHEMBL7007499

Cc1cc(C(=O)O)c(Cl)cc1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.44
NFE2L2 Q16236 1/20 0.44
ALDH1A1 P00352 1/20 0.44
TP53 P04637 1/20 0.44
TSHR P16473 1/20 0.44
CASP1 P29466 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
POLB P06746 1/20 0.43
APEX1 P27695 1/20 0.43
MYC P01106 1/20 0.42
NR4A1 P22736 1/20 0.42
CTSB P07858 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
CLCN2 P51788 2/20 0.42
ADRA2A P08913 1/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA3 P07451 1/20 0.42
CA4 P22748 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL448497 0.92 KEAP1 (0.48) KEAP1NFE2L2ALDH1A1TP53TSHR
SCHEMBL15385122 0.84 POLB (0.43) ALDH1A1TSHRSMN1; SMN2POLBAPEX1
SCHEMBL19433388 0.84 POLB (0.43) ALDH1A1TSHRSMN1; SMN2POLBAPEX1
SCHEMBL4509916 0.84 KEAP1 (0.44) KEAP1NFE2L2ALDH1A1TP53TSHR
SCHEMBL32668944 0.83 KEAP1 (0.55) KEAP1NFE2L2ALDH1A1TP53TSHR
SCHEMBL979056 0.83 KEAP1 (0.55) KEAP1NFE2L2ALDH1A1TP53TSHR
SCHEMBL3436916 0.83 KDM4E (0.45) KEAP1NFE2L2ALDH1A1LMNAHPGD
SCHEMBL10628886 0.83 ALDH1A1 (0.50) ALDH1A1TP53TSHRCASP1SMN1; SMN2
SCHEMBL14453581 0.82 CA12 (0.44) ALDH1A1TSHRCASP1SMN1; SMN2POLB
SCHEMBL364382 0.81 KEAP1 (0.48) KEAP1NFE2L2ALDH1A1TP53TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9073954-B2 5-substituted benzimidazolium compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-07-07 US disclosed
EP-0945435-B1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMA CO LTD (JP) 2003-08-13 EP disclosed
US-6136823-A BACTERICIDES OR VIRICIDES WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-0945435-A1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 1999-09-29 EP disclosed