SCHEMBL7007890

SCHEMBL7007890

COc1ccc(OC)c(S(=O)(=O)NCCCCCCNc2nsc3nccn23)c1

nearest known ligand 0.66

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
F13A1 P00488 7/20 0.66
TGM1 P22735 1/20 0.60
L3MBTL3 Q96JM7 1/20 0.49
HSD17B10 Q99714 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
ALDH1A1 P00352 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
MAPT P10636 1/20 0.46
GAA P10253 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7004379 0.91 F13A1 (0.64) F13A1TGM1SMN1; SMN2
SCHEMBL7005720 0.87 F13A1 (0.80) F13A1TGM1ALDH1A1
SCHEMBL7006472 0.86 F13A1 (0.70) F13A1TGM1ALDH1A1
SCHEMBL7008014 0.81 F13A1 (0.62) F13A1TGM1ALDH1A1
SCHEMBL7008678 0.80 F13A1 (1.00) F13A1TGM1ALDH1A1
SCHEMBL7004356 0.80 F13A1 (0.75) F13A1TGM1
SCHEMBL7014440 0.79 F13A1 (0.80) F13A1TGM1ALDH1A1SMN1; SMN2
SCHEMBL7003653 0.79 F13A1 (0.73) F13A1TGM1L3MBTL1SMN1; SMN2MAPT
SCHEMBL7004829 0.79 F13A1 (0.76) F13A1TGM1
SCHEMBL7004031 0.78 F13A1 (0.67) F13A1TGM1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030225007-A1 Sulfonamide derivatives of 3-substituted imidazol[1,2-d]-1,2,4-thiadiazoles and 3-substituted-[1,2,4] thiadiazolo[4,5-a] benzimidazole as inhibitors of fibrin cross-linking and transglutaminases APOTEX INC. 2003-12-04 US disclosed
EP-1348710-A1 Sulfonamide derivatives of 3-substituted imidazo[1,2-D]-1,2,4-thiadiazoles and 3-substituted-[1,2,4]thiadiazolo[4,5-A]benzimidazole as inhibitors of fibrin cross-linking and transglutaminases Apotex Inc. (CA) 2003-10-01 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030225007-A1 Sulfonamide derivatives of 3-substituted imidazol[1,2-d]-1,2,4-thiadiazoles and 3-substituted-[1,2,4] thiadiazolo[4,5-a] benzimidazole as inhibitors of fibrin cross-linking and transglutaminases PIGS, FGB, SERPINE1 F13A1 14/4885TGM1 7/4885L3MBTL3 1948/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.