SCHEMBL7007966

SCHEMBL7007966

N#Cc1cnc(Nc2ccc(C(=O)NCCCc3ncc[nH]3)cc2)nc1N

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 19/20 0.49
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6226700 0.79 SMN1; SMN2 (0.54) NAMPTNPC1
SCHEMBL6947662 0.77 GSK3B (0.58) NAMPT
SCHEMBL7011089 0.76 NAMPT (0.65) NAMPT
SCHEMBL6952862 0.74 IGF1R (0.50) NAMPT
SCHEMBL6949387 0.72 IGF1R (0.50) NAMPT
SCHEMBL8780738 0.71 NAMPT (0.71) NAMPT
SCHEMBL6646546 0.71 NAMPT (0.56) NAMPT
SCHEMBL1499531 0.71 NAMPT (0.55) NAMPTNPC1RAB9A
SCHEMBL7004700 0.68 MAPT (0.57) NAMPTNPC1RAB9A
SCHEMBL2447886 0.66 NPC1 (0.74) NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268445-A1 4-AMINO-5-CYANO-2-ANILINO-PYRIMIDINE DERIVATIVES AND THEIR USE AS INHIBITORS OF CELL-CYCLE KINASES AstraZeneca AB (SE) 2003-01-02 EP disclosed
WO-2001072717-A1 4-AMINO-5-CYANO-2-ANILINO-PYRIMIDINE DERIVATIVES AND THEIR USE AS INHIBITORS OF CELL-CYCLE KINASES ASTRAZENECA AB (SE) 2001-10-04 WO disclosed