SCHEMBL7008374

SCHEMBL7008374

N#Cc1cccn1-c1ccc(CBr)cc1Cl

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.35
GLA P06280 1/20 0.35
HCRTR1 O43613 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
AR P10275 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9043191 0.84 LMNA (0.36) LMNAGLAHCRTR1ALDH1A1MAPT
SCHEMBL9045587 0.83 LMNA (0.35) LMNAGLAHCRTR1ALDH1A1MAPT
SCHEMBL9041668 0.79 TSHR (0.31)
SCHEMBL7008935 0.78 KDM4E (0.38) LMNAGLAHCRTR1ALDH1A1MAPT
SCHEMBL9040399 0.78 AR (0.39) LMNAGLAALDH1A1MAPTAR
SCHEMBL7006694 0.75 LMNA (0.41) LMNAGLAHCRTR1ALDH1A1MAPT
SCHEMBL9221175 0.75 GLA (0.42) LMNAGLAHCRTR1ALDH1A1MAPT
SCHEMBL27525583 0.75 LMNA (0.38) LMNAGLAHCRTR1ALDH1A1MAPT
SCHEMBL9042519 0.74 AR (0.32) AR
SCHEMBL9043602 0.71 LMNA (0.35) LMNAGLAAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1327631-A2 Fused heterocyclic compounds, their production and use as angiotensin II antagonists Takeda Chemical Industries, Ltd. (JP) 2003-07-16 EP disclosed
EP-0518033-B1 Fused heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-07-02 EP disclosed
EP-0480204-B1 Imidazole derivatives, potent and selective antagonists of angiotensin II receptor FUJISAWA PHARMACEUTICAL CO (JP) 1996-03-20 EP disclosed
US-5389641-A Fused heterocyclic compounds, having angiotensin II antagonistic activity TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-02-14 US disclosed
US-5215994-A Treating or preventing hypertension or heart failure FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-06-01 US disclosed
US-5210092-A Hypotensive agents FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-05-11 US disclosed
EP-0518033-A1 Fused heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-12-16 EP disclosed
EP-0480204-A1 Imidazole derivatives, potent and selective antagonists of angiotensin II receptor FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-04-15 EP disclosed