SCHEMBL7009324

SCHEMBL7009324

CCOC(=O)Oc1c(-c2ccncc2)c2n(c1-c1ccc(F)cc1)CCS2

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 14/20 0.44
MAPK13 O15264 2/20 0.43
MAPK12 P53778 2/20 0.43
MAPK11 Q15759 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
KDM4E B2RXH2 1/20 0.43
CYP3A4 P08684 1/20 0.43
HPGD P15428 1/20 0.43
ALOX15 P16050 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
RIPK3 Q9Y572 2/20 0.38
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
GCGR P47871 1/20 0.36
ALOX5 P09917 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7009071 0.92 MAPK14 (0.44) MAPK14MAPK13MAPK12MAPK11SMN1; SMN2
SCHEMBL6294026 0.84 MAPK14 (0.46) MAPK14MAPK13MAPK12MAPK11SMN1; SMN2
SCHEMBL6294505 0.82 MAPK14 (0.46) MAPK14MAPK13MAPK12MAPK11SMN1; SMN2
SCHEMBL7010615 0.82 MAPK14 (0.44) MAPK14RIPK3
SCHEMBL7006565 0.82 MAPK14 (0.44) MAPK14RIPK3
SCHEMBL7008081 0.81 MAPK14 (0.44) MAPK14RIPK3
SCHEMBL7009622 0.78 MAPK14 (0.48) MAPK14MAPK13MAPK12MAPK11SMN1; SMN2
SCHEMBL7008536 0.78 RIPK3 (0.45) MAPK14RIPK3
SCHEMBL7012237 0.78 RIPK3 (0.45) MAPK14RIPK3
SCHEMBL7006189 0.77 RIPK3 (0.44) MAPK14RIPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1252163-B1 4-PYRIDYL-AND 2,4-PYRIMIDINYL-SUBSTITUTED PYRROLE DERIVATIVES AND THEIR USE IN PHARMACY MERCKLE GMBH (DE) 2003-09-24 EP disclosed
EP-1252163-A2 4-PYRIDYL-AND 2,4-PYRIMIDINYL-SUBSTITUTED PYRROLE DERIVATIVES AND THEIR USE IN PHARMACY MERCKLE GMBH (DE) 2002-10-30 EP disclosed
WO-2001057042-A2 4-PYRIDYL-AND 2,4-PYRIMIDINYL-SUBSTITUTED PYRROLE DERIVATIVES AND THEIR USE IN PHARMACY MERCKLE GMBH (DE) 2001-08-09 WO disclosed