SCHEMBL7010477

SCHEMBL7010477

Cc1ccc2cccc(OCc3c(Cl)ccc(C(=O)O)c3Cl)c2n1

nearest known ligand 0.61

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BDKRB2 P30411 18/20 0.61
PTGDR2 Q9Y5Y4 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8364184 0.85 BDKRB2 (0.67) BDKRB2
SCHEMBL7007332 0.83 BDKRB2 (0.55) BDKRB2
SCHEMBL8723959 0.82 BDKRB2 (0.67) BDKRB2
SCHEMBL7746973 0.82 BDKRB2 (0.82) BDKRB2PTGDR2
Hydrochloric Acid SCHEMBL7661562 0.82 BDKRB2 (0.66) BDKRB2
SCHEMBL6936587 0.81 BDKRB2 (0.66) BDKRB2
SCHEMBL4484397 0.81 BDKRB2 (0.60) BDKRB2
SCHEMBL4058616 0.81 BDKRB2 (0.65) BDKRB2
SCHEMBL7013654 0.81 BDKRB2 (0.62) BDKRB2
SCHEMBL27348703 0.81 BDKRB2 (0.62) BDKRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861243-B1 HETEROCYCLIC COMPOUNDS AS BRADYKININ ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 2003-11-12 EP disclosed
US-6344462-B1 Heterocyclic compounds as bradykinin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-02-05 US disclosed
US-6100284-A ANTIALLERGENS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-08 US disclosed
US-6008229-A TREATING ALLERGY, INFLAMMATION, AUTOIMMUNE DISEASE, SHOCK, PAIN FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-12-28 US disclosed
EP-0861243-A1 HETEROCYCLIC COMPOUNDS AS BRADYKININ ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-09-02 EP disclosed
WO-1997011069-A1 HETEROCYCLIC COMPOUNDS AS BRADYKININ ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-03-27 WO disclosed