SCHEMBL7010501

SCHEMBL7010501

COC(=O)c1ccc(-n2c(C)ccc2C#N)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.57
HPGD P15428 4/20 0.57
KDM4E B2RXH2 4/20 0.57
PKM P14618 1/20 0.57
NPSR1 Q6W5P4 1/20 0.57
HTT P42858 5/20 0.51
MAPT P10636 3/20 0.47
MITF O75030 1/20 0.47
LMNA P02545 1/20 0.47
TDP1 Q9NUW8 3/20 0.46
POLB P06746 2/20 0.46
MEN1 O00255 1/20 0.46
APEX1 P27695 1/20 0.46
KMT2A Q03164 1/20 0.46
MYC P01106 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA12 O43570 1/20 0.42
CA7 P43166 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9043956 0.86 HTT (0.73) ALDH1A1HPGDKDM4ENPSR1HTT
SCHEMBL15714711 0.84 ALDH1A1 (0.69) ALDH1A1HPGDKDM4EPKMNPSR1
SCHEMBL7828490 0.83 ALDH1A1 (0.55) ALDH1A1HPGDKDM4EPKMNPSR1
SCHEMBL31420342 0.73 ALDH1A1 (0.50) ALDH1A1HPGDKDM4ENPSR1HTT
SCHEMBL7007409 0.73 CTSB (0.45) ALDH1A1HPGDKDM4EPKMHTT
SCHEMBL9189815 0.72 CA1 (0.55) ALDH1A1HPGDKDM4EPKMNPSR1
SCHEMBL9043535 0.71 HPGD (0.56) ALDH1A1HPGDKDM4EPKMNPSR1
Cyanate SCHEMBL28803587 0.71 CA1 (0.64) ALDH1A1HPGDKDM4EHTTMAPT
Water SCHEMBL22720573 0.71 CA1 (0.76) ALDH1A1HPGDKDM4EHTTMAPT
SCHEMBL31420293 0.70 MAPT (0.51) ALDH1A1HPGDHTTMAPTMITF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1327631-A2 Fused heterocyclic compounds, their production and use as angiotensin II antagonists Takeda Chemical Industries, Ltd. (JP) 2003-07-16 EP disclosed
EP-0518033-B1 Fused heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-07-02 EP disclosed
US-5389641-A Fused heterocyclic compounds, having angiotensin II antagonistic activity TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-02-14 US disclosed
EP-0518033-A1 Fused heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-12-16 EP disclosed