SCHEMBL7010915

SCHEMBL7010915

CCOC(=O)C(F)C(=O)c1ccc(F)c([N+](=O)[O-])c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 3/20 0.47
ITGB1 P05556 1/20 0.46
ITGA5 P08648 1/20 0.46
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 4/20 0.44
PKM P14618 2/20 0.44
MAPT P10636 2/20 0.44
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.44
CRHBP P24387 1/20 0.44
CRHR2 Q13324 1/20 0.44
LMNA P02545 2/20 0.44
KDM4E B2RXH2 1/20 0.44
POLB P06746 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
HPGD P15428 1/20 0.43
THRB P10828 1/20 0.43
PTGER4 P35408 1/20 0.42
CLPP Q16740 2/20 0.42
MITF O75030 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7007314 0.85 KMT2A (0.40) PDK1KMT2AALDH1A1PKMMAPT
SCHEMBL1305326 0.82 KMT2A (0.64) ITGB1ITGA5KMT2AALDH1A1PKM
SCHEMBL31304627 0.82 KMT2A (0.64) ITGB1ITGA5KMT2AALDH1A1PKM
SCHEMBL10830983 0.82 CES2 (0.47) KMT2AALDH1A1MAPTRAB9ASMN1; SMN2
SCHEMBL16063547 0.80 ITGB1 (0.48) ITGB1ITGA5KMT2AALDH1A1PKM
SCHEMBL10628840 0.78 HDAC1 (0.47) ALDH1A1MAPTRAB9ANPC1LMNA
SCHEMBL31373829 0.78 ITGB1 (0.46) ITGB1ITGA5KMT2AALDH1A1PKM
SCHEMBL4302375 0.78 PDK1 (0.52) PDK1ITGB1ITGA5KMT2AALDH1A1
SCHEMBL7005289 0.77 KMT2A (0.38) KMT2AALDH1A1PKMMAPTNPC1
SCHEMBL16096851 0.76 ITGB1 (0.47) ITGB1ITGA5KMT2AALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0945435-B1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMA CO LTD (JP) 2003-08-13 EP disclosed
US-6136823-A BACTERICIDES OR VIRICIDES WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-0945435-A1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 1999-09-29 EP disclosed