SCHEMBL7010948

SCHEMBL7010948

COc1ccc(Cl)c(Oc2c(COCCOC(=O)Oc3ccsc3)nc(N3CCOCC3)nc2NS(=O)(=O)c2ccc(C(C)(C)C)cc2)c1

nearest known ligand 0.64

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 13/20 0.64
EDNRB P24530 12/20 0.47
CCR9 P51686 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7949278 0.92 EDNRA (0.64) EDNRAEDNRBCCR9
SCHEMBL7013111 0.87 EDNRA (0.80) EDNRAEDNRB
SCHEMBL7012947 0.86 EDNRA (0.48) EDNRAEDNRB
SCHEMBL7006427 0.84 EDNRA (0.81) EDNRAEDNRBCCR9
SCHEMBL7006902 0.82 EDNRA (0.70) EDNRAEDNRBCCR9
SCHEMBL7008278 0.82 EDNRA (0.70) EDNRAEDNRBCCR9
SCHEMBL7006905 0.82 EDNRA (0.70) EDNRAEDNRBCCR9
SCHEMBL7009309 0.82 EDNRA (0.76) EDNRAEDNRBCCR9
SCHEMBL9157048 0.82 EDNRA (0.73) EDNRAEDNRB
SCHEMBL7099116 0.80 EDNRA (0.63) EDNRAEDNRBCCR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0601386-B1 Sulphonamides HOFFMANN LA ROCHE (CH) 2003-02-05 EP claimed
EP-0601386-A1 Sulphonamides F. HOFFMANN-LA ROCHE AG (CH) 1994-06-15 EP claimed
EP-0601386-B1 Sulphonamides HOFFMANN LA ROCHE (CH) 2003-02-05 EP disclosed
EP-0601386-A1 Sulphonamides F. HOFFMANN-LA ROCHE AG (CH) 1994-06-15 EP disclosed