SCHEMBL7011965

SCHEMBL7011965

CCOC(=O)c1cc(-c2cn(C(C)(C)C)c3ncnc(N)c23)ccc1Oc1cccc(Cl)c1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDR P35968 9/20 0.54
LCK P06239 7/20 0.54
TEK Q02763 7/20 0.54
SRC P12931 9/20 0.51
EGFR P00533 5/20 0.45
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
JAK2 O60674 1/20 0.41
JAK3 P52333 1/20 0.41
ABL1 P00519 4/20 0.40
ABL2 P42684 4/20 0.40
EIF2AK2 P19525 1/20 0.40
EIF2AK1 Q9BQI3 1/20 0.40
EIF2AK3 Q9NZJ5 1/20 0.40
RET P07949 2/20 0.40
HCK P08631 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8128260 0.93 KDR (0.51) KDRLCKTEKSRCEGFR
SCHEMBL7011523 0.91 KDR (0.63) KDRLCKTEKSRCEGFR
SCHEMBL7007578 0.90 KDR (0.59) KDRLCKTEKSRCEGFR
SCHEMBL7014152 0.86 KDR (0.54) KDRLCKTEKSRCEGFR
SCHEMBL7010879 0.86 KDR (0.54) KDRLCKTEKSRCEGFR
SCHEMBL7013873 0.85 KDR (0.63) KDRLCKTEKSRCEGFR
SCHEMBL7007563 0.84 KDR (0.62) KDRLCKTEKSRCEGFR
SCHEMBL7012365 0.84 KDR (0.64) KDRLCKTEKSRCEGFR
SCHEMBL7005538 0.83 KDR (0.65) KDRLCKTEKSRCEGFR
SCHEMBL7004833 0.83 KDR (0.62) KDRLCKTEKSRCEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970084-B1 PYRROLO 2,3D]PYRIMIDINES AND THEIR USE AS TYROSINE KINASE INHIBITORS BASF AG (DE) 2003-06-04 EP disclosed
US-6001839-A Substituted 4-amino-7H-pyrrolo [2,3,-d]-pyrimidines as PTK inhibitors BASF AKTIENGESELLSCHAFT (DE) 1999-12-14 US disclosed