SCHEMBL7012160

SCHEMBL7012160

COc1cc(Nc2ccnc3cc(Br)ccc23)c(Cl)cc1Cl

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 9/20 0.73
GAK O14976 8/20 0.63
RIPK2 O43353 4/20 0.53
EGFR P00533 4/20 0.53
NOD1 Q9Y239 1/20 0.53
ALK Q9UM73 1/20 0.52
COQ8A Q8NI60 3/20 0.51
NLK Q9UBE8 3/20 0.51
ABL1 P00519 3/20 0.51
EPHB6 O15197 2/20 0.51
ACVR1 Q04771 2/20 0.51
STK16 O75716 1/20 0.51
AAK1 Q2M2I8 1/20 0.51
BCR P11274 1/20 0.45
POLB P06746 1/20 0.45
THRB P10828 1/20 0.45
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7015603 0.85 SRC (0.73) SRCGAKRIPK2EGFRNOD1
SCHEMBL7014373 0.81 SRC (0.67) SRCGAKRIPK2EGFRNOD1
SCHEMBL7015262 0.81 SRC (0.66) SRCGAKRIPK2EGFRNOD1
SCHEMBL5502139 0.81 SRC (0.81) SRCGAKRIPK2EGFRNOD1
SCHEMBL19617953 0.81 SRC (0.81) SRCGAKRIPK2EGFRNOD1
SCHEMBL19209424 0.81 SRC (0.81) SRCGAKRIPK2EGFRNOD1
SCHEMBL7008456 0.80 SRC (0.67) SRCGAKALDH1A1MAPT
SCHEMBL26086336 0.79 GAK (0.65) SRCGAKRIPK2EGFRALK
SCHEMBL7016099 0.78 SRC (0.61) SRCGAKALKPOLBTHRB
SCHEMBL26087214 0.78 GAK (0.63) SRCGAKRIPK2EGFRALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268431-A1 3-CYANOQUINOLINES,3-CYANO-1,6-NAPHTHYRIDINES, AND 3-CYANO-1,7-NAPHTHYRIDINES AS PROTEIN KINASE INHIBITORS Wyeth (US) 2003-01-02 EP disclosed
WO-2001072711-A1 3-CYANOQUINOLINES,3-CYANO-1,6-NAPHTHYRIDINES, AND 3-CYANO-1,7-NAPHTHYRIDINES AS PROTEIN KINASE INHIBITORS WYETH (US) 2001-10-04 WO disclosed