SCHEMBL7012232

SCHEMBL7012232

CCCC[Sn](CCCC)(CCCC)c1ccc(C#N)c(C)c1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.36
AR P10275 6/20 0.35
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
ABCG2 Q9UNQ0 1/20 0.32
MRGPRX4 Q96LA9 1/20 0.31
EGLN2 Q96KS0 1/20 0.30
IDH1 O75874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9857499 0.75 GRIN2B (0.35) TSHR
SCHEMBL1453582 0.74 TSHR (0.46) TSHRALDH1A1HPGD
SCHEMBL2389905 0.72 DRD2 (0.43) TSHR
SCHEMBL1983658 0.72 TSHR (0.32) TSHR
SCHEMBL3914612 0.71 SKP2 (0.56) TSHRARALDH1A1HPGD
SCHEMBL9901980 0.71 BDKRB2 (0.35)
SCHEMBL3790911 0.70 MYC (0.33) ALDH1A1HPGDABCG2
SCHEMBL2656551 0.70 AR (0.40) ARALDH1A1HPGD
SCHEMBL31200955 0.69 TSHR (0.40) TSHRARALDH1A1HPGD
SCHEMBL1452840 0.69 HTT (0.38) TSHRALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775702-B1 NOVEL QUINOLONE- OR NAPHTHYRIDONECARBOXYLIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO LTD (JP) 2003-07-23 EP disclosed
US-5935952-A ANTIBACTERIAL AGENT TOYAMA CHEMICAL CO., LTD. (JP) 1999-08-10 US disclosed
EP-0775702-A1 NOVEL QUINOLONE- OR NAPHTHYRIDONECARBOXYLIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 1997-05-28 EP disclosed