SCHEMBL7013216

SCHEMBL7013216

CN1CCNCC1c1ccsc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 2/20 0.34
HSD17B10 Q99714 2/20 0.33
TSHR P16473 1/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
HTR2A P28223 2/20 0.32
HTR2C P28335 2/20 0.32
HTR2B P41595 2/20 0.32
CHRNB2 P17787 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA7 P36544 1/20 0.31
CHRNA4 P43681 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3976295 0.76 CHRNB2 (0.55) HPGDTAAR1HTR2AHTR2CHTR2B
SCHEMBL1579434 0.76 CHRNB2 (0.55) HPGDTAAR1HTR2AHTR2CHTR2B
SCHEMBL18913839 0.76 CHRNB2 (0.55) HPGDTAAR1HTR2AHTR2CHTR2B
SCHEMBL470846 0.76 CHRNB2 (0.55) HPGDTAAR1HTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL27673502 0.75 CHRNB2 (0.53) HPGDTAAR1HTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL1722775 0.75 CHRNB2 (0.53) HPGDTAAR1HTR2AHTR2CHTR2B
SCHEMBL13162098 0.75 CHRNB2 (0.58) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL6026785 0.75 ADRB1 (0.43) HTR2CCHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL5734703 0.75 KDM4E (0.41) KDM4EGAAHTR2CHTR2B
SCHEMBL7400548 0.73 MAOB (0.39) HTR2AHTR2CHTR2BCHRNB2CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1419545-A 3-cyanoquinolines, 3-cyano-1,6-naphthyridines, and 3-cyano-1,7-naphthyridines as protein kinase inhibitors WYETH CORP (US) 2003-05-21 CN disclosed
EP-1268431-A1 3-CYANOQUINOLINES,3-CYANO-1,6-NAPHTHYRIDINES, AND 3-CYANO-1,7-NAPHTHYRIDINES AS PROTEIN KINASE INHIBITORS Wyeth (US) 2003-01-02 EP disclosed
WO-2001072711-A1 3-CYANOQUINOLINES,3-CYANO-1,6-NAPHTHYRIDINES, AND 3-CYANO-1,7-NAPHTHYRIDINES AS PROTEIN KINASE INHIBITORS WYETH (US) 2001-10-04 WO disclosed