SCHEMBL7013628

SCHEMBL7013628

COCc1cc[c]c(C(N)=O)n1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.34
CDK8 P49336 1/20 0.32
CDK19 Q9BWU1 1/20 0.32
NNMT P40261 2/20 0.32
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
POLB P06746 2/20 0.31
TSHR P16473 1/20 0.31
CASP1 P29466 1/20 0.31
HSD17B10 Q99714 1/20 0.31
ADORA2A P29274 2/20 0.31
ADORA1 P30542 2/20 0.31
ADORA3 P0DMS8 1/20 0.30
ADORA2B P29275 1/20 0.30
NTRK1 P04629 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
PARP1 P09874 1/20 0.30
PARP10 Q53GL7 1/20 0.30
PARP2 Q9UGN5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4261549 0.80
SCHEMBL3197756 0.80 CCR1 (0.36)
SCHEMBL3211526 0.77 PARP1 (0.35) PARP1PARP2
SCHEMBL3315095 0.75 HPGD (0.37) HRH3POLBPARP1PARP2
SCHEMBL2791847 0.75 NNMT (0.49) NNMTPOLBCA1CA2PARP1
SCHEMBL2794698 0.74 IKBKB (0.37) NNMTTSHRCA1CA2
SCHEMBL3114993 0.72 PARP1 (0.43) NNMTPOLBPARP1
SCHEMBL2791507 0.72 HCAR3 (0.44) HSD17B10
SCHEMBL3002690 0.71 PIM1 (0.39) NNMTLMNAPOLBTSHRCASP1
SCHEMBL6309563 0.71 PARP10 (0.41) NNMTTSHRPARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1325006-A2 HETEROCYCLIC COMPOUNDS AS LIGANDS OF THE GABA A? RECEPTOR NEUROGEN CORPORATION (US) 2003-07-09 EP claimed
WO-2002012442-A2 HETEROCYCLIC COMPOUNDS AS LIGANDS OF THE GABAA RECEPTOR NEUROGEN CORPORATION (US) 2002-02-14 WO claimed