SCHEMBL7014222

SCHEMBL7014222

COc1cccc(CC#Cc2cn3c(=O)n(Cc4ccc(S)cc4)c(=O)c(C)c3s2)c1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 11/20 0.41
THRB P10828 3/20 0.40
MAPT P10636 2/20 0.40
ALDH1A1 P00352 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
LMNA P02545 2/20 0.38
TP53 P04637 1/20 0.38
CMA1 P23946 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5957762 0.93 TRPA1 (0.48) TRPA1THRBMAPTALDH1A1L3MBTL1
SCHEMBL5957317 0.91 TRPA1 (0.41) TRPA1THRBMAPTALDH1A1L3MBTL1
SCHEMBL5957855 0.90 TRPA1 (0.42) TRPA1THRBMAPTALDH1A1L3MBTL1
SCHEMBL5957416 0.90 TRPA1 (0.40) TRPA1THRBMAPTALDH1A1L3MBTL1
SCHEMBL5957381 0.89 TRPA1 (0.45) TRPA1THRBMAPTLMNATP53
SCHEMBL5957451 0.89 TRPA1 (0.45) TRPA1
SCHEMBL5957508 0.88 TRPA1 (0.39) TRPA1THRBMAPTALDH1A1L3MBTL1
SCHEMBL5957619 0.87 TRPA1 (0.39) TRPA1THRBMAPTALDH1A1L3MBTL1
SCHEMBL5957812 0.85 TRPA1 (0.44) TRPA1THRBMAPTLMNA
SCHEMBL5957672 0.84 CXCR3 (0.43) TRPA1THRBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362054-A1 BICYCLIC PYRIMIDINE MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2003-11-19 EP claimed
WO-2002064599-A1 BICYCLIC PYRIMIDINE MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2002-08-22 WO claimed