SCHEMBL7014392

SCHEMBL7014392

COC(=O)C(C)c1ccc(-c2cncc(Br)c2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.47
XDH P47989 3/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
LMNA P02545 2/20 0.41
GAA P10253 2/20 0.41
HPGD P15428 2/20 0.41
ALDH1A1 P00352 2/20 0.39
MAPT P10636 2/20 0.39
MAPK1 P28482 2/20 0.39
TP53 P04637 1/20 0.39
MT-CO2 P00403 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
PTGS1 P23219 1/20 0.39
MAP4K4 O95819 1/20 0.39
CYP2A6 P11509 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL749046 0.82 PTGS1 (0.41) PTGS2MEN1KMT2ALMNAGAA
SCHEMBL7009837 0.79 PTGS2 (0.75) PTGS2XDHHPGDMT-CO2MKNK1
SCHEMBL7009835 0.79 PTGS2 (0.75) PTGS2XDHHPGDMT-CO2MKNK1
SCHEMBL4901239 0.77 CYP2A6 (0.47) PTGS2MEN1KMT2ALMNAGAA
SCHEMBL5148090 0.77 CYP1A2 (0.51) PTGS2KMT2AHPGDALDH1A1MT-CO2
SCHEMBL22554086 0.77 CYP11B1 (0.51) XDHMEN1KMT2AALDH1A1MAPT
SCHEMBL3729385 0.75 PTGS2 (0.58) PTGS2KMT2AHPGDMT-CO2PTGS1
SCHEMBL3672641 0.75 CTSK (0.41) XDHMEN1KMT2ALMNAGAA
SCHEMBL4162120 0.75 CTSK (0.41) XDHMEN1KMT2ALMNAGAA
SCHEMBL4154310 0.75 CTSK (0.41) XDHMEN1KMT2ALMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054857-B1 BIARYL-ACETIC ACID DERIVATIVES AND THEIR USE AS COX-2 INHIBITORS MERCK FROSST CANADA INC (CA) 2003-11-05 EP disclosed
US-5994379-A Bisaryl COX-2 inhibiting compounds, compositions and methods of use MERCK FROSST CANADA, INC. (CA) 1999-11-30 US disclosed