SCHEMBL7014397

SCHEMBL7014397

Cn1c(SCc2ccc(C(=O)c3ccc(Cl)cc3)cc2)nc2ccc(O)cc2c1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.50
TP53 P04637 1/20 0.50
THRB P10828 1/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
LMNA P02545 1/20 0.46
DRD2 P14416 2/20 0.45
TBXA2R P21731 2/20 0.45
TDP1 Q9NUW8 1/20 0.45
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7013210 0.93 MEN1 (0.53) MAPTTP53THRBMEN1KMT2A
SCHEMBL7019775 0.90 MEN1 (0.58) MAPTTP53THRBMEN1KMT2A
SCHEMBL7020177 0.90 MAPT (0.54) MAPTTP53THRBMEN1KMT2A
SCHEMBL7014022 0.89 MEN1 (0.46) MAPTTP53THRBMEN1KMT2A
SCHEMBL7012409 0.88 HDAC3 (0.54) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7011327 0.87 MEN1 (0.47) MAPTTP53THRBMEN1KMT2A
SCHEMBL7017207 0.87 HDAC3 (0.56) MAPTTP53THRBCYP1A2CYP2D6
SCHEMBL7015339 0.86 KMT2A (0.68) MAPTTP53MEN1KMT2ACYP1A2
SCHEMBL7017745 0.85 MAPT (0.47) MAPTTP53THRBMEN1KMT2A
SCHEMBL7021244 0.84 MEN1 (0.54) MEN1KMT2ANPSR1HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed