SCHEMBL7015339

SCHEMBL7015339

Cn1c(SCc2ccc(C(=O)c3ccc(Cl)cc3)cc2)nc2ccccc2c1=O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.68
MEN1 O00255 2/20 0.68
CYP1A2 P05177 1/20 0.63
CYP2D6 P10635 1/20 0.63
MAPT P10636 1/20 0.63
CYP2C9 P11712 1/20 0.63
CYP2C19 P33261 1/20 0.63
NPSR1 Q6W5P4 1/20 0.63
USP2 O75604 1/20 0.59
TDP1 Q9NUW8 1/20 0.58
DRD2 P14416 2/20 0.55
TBXA2R P21731 2/20 0.55
L3MBTL1 Q9Y468 2/20 0.54
CA12 O43570 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA9 Q16790 1/20 0.54
TP53 P04637 1/20 0.53
PTGDR2 Q9Y5Y4 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7018117 0.91 TDP1 (0.64) KMT2AMEN1CYP1A2CYP2D6MAPT
SCHEMBL7013706 0.89 KMT2A (0.68) KMT2AMEN1MAPTUSP2TDP1
SCHEMBL7013210 0.89 MEN1 (0.53) KMT2AMEN1CYP1A2CYP2D6MAPT
SCHEMBL7015464 0.89 KMT2A (0.60) KMT2AMEN1CYP1A2CYP2D6MAPT
SCHEMBL8646764 0.87 L3MBTL1 (0.68) KMT2AMEN1CYP1A2CYP2D6MAPT
SCHEMBL7019775 0.86 MEN1 (0.58) KMT2AMEN1CYP1A2CYP2D6MAPT
SCHEMBL7014397 0.86 MAPT (0.50) KMT2AMEN1CYP1A2CYP2D6MAPT
SCHEMBL7014308 0.85 DRD2 (0.59) KMT2AMEN1CYP1A2CYP2D6MAPT
SCHEMBL7011002 0.85 MEN1 (0.48) KMT2AMEN1CYP1A2CYP2D6MAPT
SCHEMBL7507339 0.85 MEN1 (0.56) KMT2AMEN1CYP1A2CYP2D6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed