SCHEMBL7019775

SCHEMBL7019775

Cc1ccc2nc(SCc3ccc(C(=O)c4ccc(Cl)cc4)cc3)n(C)c(=O)c2c1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.58
KMT2A Q03164 1/20 0.58
TDP1 Q9NUW8 1/20 0.53
MAPT P10636 2/20 0.50
TP53 P04637 1/20 0.50
THRB P10828 1/20 0.50
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7013210 0.93 MEN1 (0.53) MEN1KMT2ATDP1MAPTTP53
SCHEMBL7014397 0.90 MAPT (0.50) MEN1KMT2ATDP1MAPTTP53
SCHEMBL7017207 0.87 HDAC3 (0.56) MAPTTP53THRBCYP1A2CYP2D6
SCHEMBL7015339 0.86 KMT2A (0.68) MEN1KMT2ATDP1MAPTTP53
SCHEMBL7017745 0.85 MAPT (0.47) MEN1KMT2AMAPTTP53THRB
SCHEMBL7021244 0.84 MEN1 (0.54) MEN1KMT2ANPSR1
SCHEMBL7507339 0.82 MEN1 (0.56) MEN1KMT2ATDP1MAPTTP53
SCHEMBL9060596 0.81 MAOA (0.52) MEN1KMT2AMAPTTP53THRB
SCHEMBL7015444 0.80 HDAC3 (0.59) MEN1KMT2A
SCHEMBL7018117 0.80 TDP1 (0.64) MEN1KMT2ATDP1MAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed