Bicarbonate

Bicarbonate

SCHEMBL7014535

CCc1cc2c(NCc3cccc([N+](=O)[O-])c3)nc(C3CCCCC3)nc2s1.O=C(O)O

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 3/20 0.44
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 2/20 0.44
POLB P06746 2/20 0.43
ICAM1 P05362 1/20 0.41
SELE P16581 1/20 0.41
VCAM1 P19320 1/20 0.41
MAPT P10636 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
HSD17B10 Q99714 1/20 0.38
KCNN3 Q9UGI6 1/20 0.38
VCP P55072 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8179882 0.91 PDE5A (0.43) PDE5AALDH1A1KDM4EPOLBICAM1
Bicarbonate SCHEMBL7018952 0.90 PDE5A (0.46) PDE5AALDH1A1KDM4EPOLBMAPT
Bicarbonate SCHEMBL7014883 0.89 PDE5A (0.46) PDE5AALDH1A1KDM4EPOLBMAPT
Bicarbonate SCHEMBL7015579 0.88 PDE5A (0.46) PDE5AALDH1A1KDM4EPOLBMAPT
Bicarbonate SCHEMBL7016629 0.88 PDE5A (0.57) PDE5AALDH1A1KDM4EICAM1SELE
Bicarbonate SCHEMBL7009687 0.88 PDE5A (0.43) PDE5AALDH1A1KDM4EPOLBMAPT
SCHEMBL7422996 0.84 PDE5A (0.61) PDE5AALDH1A1KDM4EICAM1SELE
Bicarbonate SCHEMBL7021386 0.83 ALDH1A1 (0.47) PDE5AALDH1A1KDM4EPOLBMAPT
Bicarbonate SCHEMBL7011757 0.82 ACHE (0.44) PDE5AALDH1A1KDM4EICAM1SELE
Bicarbonate SCHEMBL7013925 0.82 PDE5A (0.43) PDE5AALDH1A1KDM4EICAM1SELE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934321-B1 THIENOPYRIMIDINE WITH PHOSPHODIESTERASE V INHIBITING EFFECT MERCK PATENT GMBH (DE) 2003-08-06 EP disclosed