SCHEMBL7014540

SCHEMBL7014540

CCn1c(SCc2ccc(C(=O)c3ccc(Cl)cc3)cc2)nc2cccc(C)c2c1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.52
TBXA2R P21731 7/20 0.52
HDAC3 O15379 2/20 0.48
HDAC4 P56524 2/20 0.48
HDAC1 Q13547 2/20 0.48
HDAC7 Q8WUI4 2/20 0.48
HDAC2 Q92769 2/20 0.48
HDAC10 Q969S8 2/20 0.48
HDAC11 Q96DB2 2/20 0.48
HDAC8 Q9BY41 2/20 0.48
HDAC6 Q9UBN7 2/20 0.48
HDAC9 Q9UKV0 2/20 0.48
HDAC5 Q9UQL6 2/20 0.48
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48
PTGDR2 Q9Y5Y4 1/20 0.48
TP53 P04637 4/20 0.47
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7017988 0.90 MEN1 (0.61) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7017497 0.89 TDP1 (0.52) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7018370 0.88 MEN1 (0.50) DRD2TBXA2RHDAC3HDAC4HDAC1
SCHEMBL7015553 0.88 MEN1 (0.48) DRD2TBXA2RHDAC3HDAC4HDAC1
SCHEMBL7011506 0.82 MEN1 (0.55) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7018222 0.81 TDP1 (0.49) DRD2TBXA2RKMT2AMEN1PTGDR2
SCHEMBL7017586 0.80 MEN1 (0.57) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7101327 0.80 MEN1 (0.60) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7014213 0.79 DRD2 (0.48) DRD2TBXA2RHDAC3HDAC4HDAC1
SCHEMBL7014429 0.79 MEN1 (0.54) DRD2TBXA2RHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed