SCHEMBL7014670

SCHEMBL7014670

CC(=O)Nc1ccc2s[nH]c(=O)c2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
G6PD P11413 2/20 0.49
KDM4E B2RXH2 4/20 0.48
ALDH1A1 P00352 3/20 0.48
ESR1 P03372 1/20 0.48
HPGD P15428 1/20 0.48
MTNR1A P48039 2/20 0.47
MTNR1B P49286 2/20 0.47
KMT2A Q03164 2/20 0.47
ERCC1 P07992 1/20 0.46
DNASE1 P24855 1/20 0.46
FEN1 P39748 1/20 0.46
ERCC4 Q92889 1/20 0.46
PSMB8 P28062 1/20 0.46
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
MAOA P21397 2/20 0.43
MAPT P10636 2/20 0.43
DDAH1 O94760 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL79222 0.88 ALDH1A1 (0.50) G6PDKDM4EALDH1A1ESR1HPGD
SCHEMBL18122812 0.80 ALDH1A1 (0.49) KDM4EALDH1A1HPGDKMT2AMAPT
SCHEMBL11540003 0.79 KDM4E (0.51) G6PDKDM4EALDH1A1ESR1HPGD
SCHEMBL4869324 0.76 KDM4E (0.54) G6PDKDM4EALDH1A1ESR1HPGD
SCHEMBL3868022 0.71 MAPT (0.53) KDM4EALDH1A1HPGDKMT2AMAOA
SCHEMBL5106815 0.70 MAPT (0.65) G6PDKDM4EALDH1A1HPGDMTNR1A
SCHEMBL12922996 0.70 PFKFB3 (0.53) G6PDKDM4EALDH1A1ESR1HPGD
SCHEMBL22281315 0.70 KDM4E (0.68) G6PDKDM4EALDH1A1HPGDMTNR1A
SCHEMBL15237053 0.70 ALDH1A1 (0.67) G6PDKDM4EALDH1A1ESR1HPGD
SCHEMBL12278579 0.69 LDHA (0.57) G6PDKDM4EALDH1A1KMT2APSMB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828488-B1 ISOTHIAZOLONES WARNER LAMBERT CO (US) 2003-02-12 EP claimed
EP-0828488-A1 ISOTHIAZOLONES WARNER-LAMBERT COMPANY (US) 1998-03-18 EP claimed
WO-1996038144-A1 ISOTHIAZOLONES WARNER-LAMBERT COMPANY (US) 1996-12-05 WO claimed
CN-1114402-C Isothiazolones WARNER LAMBERT CO (US) 2003-07-16 CN disclosed
EP-0828488-B1 ISOTHIAZOLONES WARNER LAMBERT CO (US) 2003-02-12 EP disclosed
US-6133270-A Isothiazolones and pharmaceutical formulations WARNER-LAMBERT COMPANY (US) 2000-10-17 US disclosed
US-6001863-A USEFUL AS ANTIVIRAL, ANTIINFLAMMATORY AND ANTIATHEROSCLEROSIS AGENT; ADMINISTERING TO THE PATIENT IN NEED OF ZINC EJECTION FROM NUCLEOCAPSID PROTEIN WARNER-LAMBERT COMPANY (US) 1999-12-14 US disclosed
US-5889034-A ANTIINFLAMMATORY AGENT; ANTIATHEROSCLEROSIS AGENT; VIRICIDES WARNER-LAMBERT COMPANY (US) 1999-03-30 US disclosed
US-5733921-A ANTIRETROVIRAL AGENTS; ANTIINFLAMMATORY AGENTS; ANTIATHEROSCLEROSIS WARNER-LAMBERT COMPANY (US) 1998-03-31 US disclosed
US-5668162-A Isothiazolones lower plasma levels of lipoprotein(a) WARNER-LAMBERT COMPANY 1997-09-16 US disclosed
US-5620997-A VIRICIDES, ANTIINFLAMMATORY AGENTS, ANTIATHEROSCLEROTIC AGENT WARNER-LAMBERT COMPANY (US) 1997-04-15 US disclosed