SCHEMBL7015177

SCHEMBL7015177

COc1ccc2nccc([C@H](CO)N3CCC(CO)(NCc4cc5ccccc5o4)CC3)c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR8 P51685 1/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
GAA P10253 1/20 0.41
SLC2A1 P11166 2/20 0.37
HTR2B P41595 4/20 0.37
HTR1A P08908 3/20 0.37
DRD2 P14416 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
KCNH2 Q12809 2/20 0.36
CYP2D6 P10635 5/20 0.35
KDM4E B2RXH2 4/20 0.35
ALDH1A1 P00352 3/20 0.35
HPGD P15428 3/20 0.35
HSD17B10 Q99714 3/20 0.35
TSHR P16473 1/20 0.35
CYP3A4 P08684 1/20 0.35
CHRM2 P08172 1/20 0.35
ADRA2A P08913 1/20 0.35
SLC6A4 P31645 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4275487 0.88 SLC2A1 (0.48) CCR8MEN1KMT2AGAASLC2A1
SCHEMBL5652075 0.78 CCR8 (0.45) CCR8MEN1KMT2ASLC2A1HTR2B
SCHEMBL4275508 0.73 KCNH2 (0.65) CCR8SLC2A1KCNH2
SCHEMBL5778069 0.73 MEN1 (0.38) MEN1KMT2AGAASLC2A1HTR2B
SCHEMBL6985392 0.72 NCF1 (0.58) MEN1KMT2AHTR2BHTR1ADRD2
SCHEMBL7017484 0.71 CYP2D6 (0.48) MEN1KMT2ASLC2A1HTR2BDRD2
SCHEMBL3690599 0.70 KCNH2 (0.50) CCR8MEN1KMT2ASLC2A1KCNH2
SCHEMBL6988402 0.69 CYP2D6 (0.44) MEN1KMT2ASLC2A1HTR2BDRD2
SCHEMBL13145896 0.69 KCNH2 (0.48) CCR8MEN1KMT2ASLC2A1HTR2B
SCHEMBL7146164 0.68 SLC2A1 (0.48) MEN1KMT2ASLC2A1DRD2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1305308-A1 AMINOPIPERIDINE QUINOLINES AND THEIR AZAISOSTERIC ANALOGUES WITH ANTIBACTERIAL ACTIVITY SMITHKLINE BEECHAM PLC (GB) 2003-05-02 EP disclosed
WO-2002008224-A1 AMINOPIPERIDINE QUINOLINES AND THEIR AZAISOSTERIC ANALOGUES WITH ANTIBACTERIAL ACTIVITY SMITHKLINE BEECHAM P.L.C. (GB) 2002-01-31 WO disclosed