SCHEMBL7015293

SCHEMBL7015293

COc1ccc(CNc2nc(N3CCC(OC(=O)O)CC3)nc3sc(C)c(C)c23)cc1OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.41
GAA P10253 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
PDE5A O76074 2/20 0.40
NPC1 O15118 1/20 0.40
NR2F2 P24468 1/20 0.40
RAB9A P51151 1/20 0.40
EPHX2 P34913 1/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
LMNA P02545 2/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ACHE P22303 4/20 0.38
APP P05067 4/20 0.38
BCHE P06276 1/20 0.38
CCR4 P51679 1/20 0.37
CHRM5 P08912 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7020191 0.93 PDE5A (0.48) PDE5A
SCHEMBL7019915 0.93 PDE5A (0.42) TP53PDE5AAPPCCR4
SCHEMBL7016681 0.91 KDM4E (0.40) TP53GAARXFP1PDE5ANPC1
SCHEMBL8179618 0.90 PDE4A (0.44) TP53GAARXFP1PDE5ANPC1
SCHEMBL7020121 0.88 GAA (0.41) GAARXFP1PDE5AALDH1A1KDM4E
SCHEMBL7012724 0.88 GAA (0.45) GAARXFP1ALDH1A1KDM4ELMNA
SCHEMBL7012162 0.87 ALDH1A1 (0.44) GAARXFP1PDE5ARAB9AEPHX2
SCHEMBL7018507 0.87 PDE5A (0.48) PDE5A
SCHEMBL7022471 0.87 TP53 (0.41) TP53PDE5ASMN1; SMN2ACHEAPP
SCHEMBL7013924 0.87 MAPT (0.45) TP53GAAALDH1A1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934321-B1 THIENOPYRIMIDINE WITH PHOSPHODIESTERASE V INHIBITING EFFECT MERCK PATENT GMBH (DE) 2003-08-06 EP disclosed