SCHEMBL7015329

SCHEMBL7015329

COC(=O)c1cccc(C(=O)CC#N)c1F

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.54
KDM4E B2RXH2 5/20 0.54
HSD17B10 Q99714 3/20 0.54
KMT2A Q03164 5/20 0.43
MEN1 O00255 3/20 0.43
POLB P06746 2/20 0.42
ATM Q13315 1/20 0.42
MAPT P10636 3/20 0.42
LMNA P02545 2/20 0.41
TSHR P16473 2/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
CFTR P13569 1/20 0.40
MRGPRX4 Q96LA9 1/20 0.39
GLA P06280 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
KCNH2 Q12809 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7012838 0.84 NPC1 (0.43) ALDH1A1KDM4EHSD17B10KMT2AMEN1
SCHEMBL28539594 0.84 KDM4E (0.63) ALDH1A1KDM4EHSD17B10KMT2AMEN1
SCHEMBL1401560 0.82 TSHR (0.57) ALDH1A1KDM4EHSD17B10KMT2AMEN1
SCHEMBL22579325 0.80 ALDH1A1 (0.47) ALDH1A1KDM4EHSD17B10KMT2AMEN1
SCHEMBL17479435 0.80 PTPN1 (0.45) ALDH1A1KDM4EHSD17B10KMT2APOLB
SCHEMBL12694512 0.80 MAPT (0.46) ALDH1A1KDM4EHSD17B10KMT2AMEN1
SCHEMBL31438543 0.80 PTPN1 (0.45) ALDH1A1KDM4EHSD17B10KMT2APOLB
SCHEMBL3563696 0.79 CES2 (0.55) ALDH1A1KDM4EHSD17B10KMT2AMEN1
SCHEMBL4968519 0.79 ALDH1A1 (0.47) ALDH1A1KDM4EHSD17B10KMT2AMEN1
SCHEMBL2134625 0.79 KDM4E (0.52) ALDH1A1KDM4EHSD17B10KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1327631-A2 Fused heterocyclic compounds, their production and use as angiotensin II antagonists Takeda Chemical Industries, Ltd. (JP) 2003-07-16 EP disclosed
EP-0518033-B1 Fused heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-07-02 EP disclosed
US-5389641-A Fused heterocyclic compounds, having angiotensin II antagonistic activity TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-02-14 US disclosed
EP-0518033-A1 Fused heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-12-16 EP disclosed