SCHEMBL7015484

SCHEMBL7015484

O=C(c1ccc(Cl)cc1)c1ccc(Cn2cnc3c(Cl)nnc(Cl)c32)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.44
P2RX7 Q99572 1/20 0.44
HDAC1 Q13547 3/20 0.43
VNN1 O95497 2/20 0.43
HDAC4 P56524 1/20 0.43
MAPK1 P28482 2/20 0.42
LMNA P02545 1/20 0.42
HDAC2 Q92769 2/20 0.40
HDAC3 O15379 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
SCD O00767 1/20 0.40
YTHDC1 Q96MU7 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
HTT P42858 1/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7016174 0.82 VNN1 (0.41) HDAC6P2RX7HDAC1VNN1HDAC4
SCHEMBL7012720 0.82 VNN1 (0.41) HDAC6P2RX7HDAC1VNN1HDAC4
SCHEMBL7012213 0.81 LMNA (0.48) HDAC6P2RX7HDAC1VNN1HDAC4
SCHEMBL7011737 0.81 LMNA (0.48) HDAC6P2RX7HDAC1VNN1HDAC4
SCHEMBL7011613 0.80 MAPK1 (0.43) HDAC6P2RX7HDAC1VNN1HDAC4
SCHEMBL7013123 0.77 HDAC1 (0.46) HDAC6HDAC1VNN1HDAC4MAPK1
SCHEMBL23462025 0.77 ADORA2A (0.48) LMNAYTHDC1SMN1; SMN2CYP11B1CYP11B2
SCHEMBL29888748 0.77 ADORA2A (0.48) LMNAYTHDC1SMN1; SMN2CYP11B1CYP11B2
SCHEMBL7009400 0.77 HDAC6 (0.41) HDAC6P2RX7HDAC1VNN1HDAC4
SCHEMBL7012335 0.73 LMNA (0.45) HDAC6HDAC1VNN1HDAC4MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed